SCHEMBL17565616

SCHEMBL17565616

C=CC[C@@H](C)[C@@H](C)S(=O)(=O)N(Cc1ccc(C)cc1)Cc1ccc(OC)cc1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
APLNR P35414 17/20 0.56
MAPT P10636 1/20 0.43
PKM P14618 1/20 0.43
CNR2 P34972 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17565620 1.00 APLNR (0.56) APLNRMAPTPKMCNR2
SCHEMBL17565619 1.00 APLNR (0.56) APLNRMAPTPKMCNR2
SCHEMBL17565617 1.00 APLNR (0.56) APLNRMAPTPKMCNR2
SCHEMBL19285603 0.95 APLNR (0.58) APLNR
SCHEMBL20630075 0.95 APLNR (0.58) APLNR
SCHEMBL17542462 0.95 APLNR (0.58) APLNR
SCHEMBL17542301 0.95 APLNR (0.58) APLNR
SCHEMBL17542133 0.95 APLNR (0.58) APLNR
SCHEMBL17542354 0.95 APLNR (0.58) APLNR
SCHEMBL17565615 0.87 APLNR (0.50) APLNRMAPTPKMCNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12024529-B2 Compounds that inhibit MCL-1 protein AMGEN INC. (US) 2024-07-02 US disclosed
US-20230271981-A1 COMPOUNDS THAT INHIBIT MCL-1 PROTEIN AMGEN INC. (US) 2023-08-31 US disclosed
US-11685747-B2 Compounds that inhibit MCL-1 protein AMGEN INC. (US) 2023-06-27 US disclosed
US-20170088560-A1 COMPOUNDS THAT INHIBIT MCL-1 PROTEIN AMGEN INC. (US) 2017-03-30 US disclosed
US-9562061-B2 Compounds that inhibit MCL-1 protein AMGEN INC. (US) 2017-02-07 US disclosed
US-20160068545-A1 COMPOUNDS THAT INHIBIT MCL-1 PROTEIN AMGEN INC. (US) 2016-03-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230271981-A1 COMPOUNDS THAT INHIBIT MCL-1 PROTEIN MCL1, BCL2L1, BCL9 APLNR 3940/4885MAPT 3369/4885PKM 3161/4885
US-11685747-B2 Compounds that inhibit MCL-1 protein MCL1, BCL2L1, BCL9 APLNR 3940/4885MAPT 3369/4885PKM 3161/4885
US-12024529-B2 Compounds that inhibit MCL-1 protein MCL1, BCL2L1, BCL9 APLNR 3940/4885MAPT 3369/4885PKM 3161/4885
US-20160068545-A1 COMPOUNDS THAT INHIBIT MCL-1 PROTEIN MCL1, BCL9, BCL2L1 APLNR 3701/4885MAPT 3153/4885PKM 3036/4885
US-20170088560-A1 COMPOUNDS THAT INHIBIT MCL-1 PROTEIN MCL1, BCL9, BCL2L1 APLNR 3701/4885MAPT 3153/4885PKM 3036/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.