SCHEMBL17568784

SCHEMBL17568784

CC(C)CC1(CCc2ccccc2)NC(=N)N(Cc2ccc(CNO)cc2)C1=O

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.45
HDAC6 Q9UBN7 4/20 0.42
ATM Q13315 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.36
ELANE P08246 2/20 0.36
THRB P10828 1/20 0.35
IDO1 P14902 1/20 0.35
CYP2C19 P33261 2/20 0.35
CNR1 P21554 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 1/20 0.34
FPR2 P25090 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7516869 0.91 BACE1 (0.55) BACE1HDAC6ATML3MBTL1MEN1
SCHEMBL8265141 0.89 BACE1 (0.49) BACE1HDAC6ATML3MBTL1MEN1
SCHEMBL17568772 0.88 BACE1 (0.42) BACE1HDAC6ATML3MBTL1ELANE
SCHEMBL7524106 0.84 BACE1 (0.67) BACE1HDAC6L3MBTL1CYP2C19
SCHEMBL13722748 0.83 BACE1 (0.50) BACE1MEN1ALDH1A1KMT2AFPR2
SCHEMBL7517002 0.81 SMN1; SMN2 (0.50) BACE1L3MBTL1MEN1ALDH1A1KMT2A
SCHEMBL7524743 0.81 BACE1 (0.58) BACE1CNR1MEN1KMT2AFPR2
SCHEMBL10305492 0.79 BACE1 (0.46) BACE1HDAC6L3MBTL1ALDH1A1
SCHEMBL7516805 0.74 BACE1 (0.47) BACE1HDAC6ATML3MBTL1ELANE
SCHEMBL7527379 0.74 BACE1 (0.51) BACE1HDAC6ATMMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2153832-B1 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2016-03-09 EP disclosed