SCHEMBL8265141

SCHEMBL8265141

CC(=O)NCc1ccc(CN2C(=N)NC(CCc3ccccc3)(CC(C)C)C2=O)cc1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 3/20 0.49
HDAC6 Q9UBN7 1/20 0.41
HTR2A P28223 3/20 0.39
HTR2C P28335 3/20 0.39
HTR2B P41595 3/20 0.39
NR3C2 P08235 1/20 0.39
ATM Q13315 1/20 0.38
PTPN1 P18031 1/20 0.37
ALDH1A1 P00352 3/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
RORC P51449 1/20 0.37
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7516869 0.94 BACE1 (0.55) BACE1HDAC6NR3C2ATMPTPN1
SCHEMBL17568784 0.89 BACE1 (0.45) BACE1HDAC6ATMALDH1A1L3MBTL1
SCHEMBL7524106 0.87 BACE1 (0.67) BACE1HDAC6L3MBTL1
SCHEMBL13722748 0.86 BACE1 (0.50) BACE1PTPN1ALDH1A1RORCKMT2A
SCHEMBL17568772 0.85 BACE1 (0.42) BACE1HDAC6ATML3MBTL1KMT2A
SCHEMBL7524743 0.84 BACE1 (0.58) BACE1NR3C2PTPN1KMT2AMEN1
SCHEMBL7517002 0.82 SMN1; SMN2 (0.50) BACE1NR3C2ALDH1A1L3MBTL1KMT2A
SCHEMBL10305492 0.82 BACE1 (0.46) BACE1HDAC6NR3C2PTPN1ALDH1A1
SCHEMBL7516414 0.80 BACE1 (0.42) BACE1HDAC6ALDH1A1KMT2AMAPT
SCHEMBL7516805 0.79 BACE1 (0.47) BACE1HDAC6NR3C2ATMPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1838304-B1 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS SCHERING CORP (US) 2009-08-19 EP disclosed
WO-2006065277-A2 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS SCHERING CORPORATION (US) 2006-06-22 WO disclosed