SCHEMBL17568880

SCHEMBL17568880

N=C1NC(CCC2CCCCC2)(CC2CCCCC2)C(=O)N1Cc1ccc(CN2CCNC2=O)cc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 9/20 0.42
POLB P06746 2/20 0.39
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.37
MAPT P10636 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
GRM2 Q14416 4/20 0.34
CTSD P07339 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRK1 P41145 1/20 0.32
OPRL1 P41146 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7512656 0.86 ALDH1A1 (0.46) BACE1POLBALDH1A1SMN1; SMN2CTSD
SCHEMBL8289351 0.85 BACE1 (0.40) BACE1ALDH1A1SMN1; SMN2MAPTCTSD
SCHEMBL7518136 0.84 BACE1 (0.40) BACE1ALDH1A1CTSDKMT2AOPRM1
SCHEMBL7512357 0.82 ALDH1A1 (0.49) BACE1POLBALDH1A1SMN1; SMN2MAPT
SCHEMBL7512798 0.82 BACE1 (0.40) BACE1CTSDMEN1OPRM1OPRL1
SCHEMBL7513207 0.82 BACE1 (0.37) BACE1CTSDKMT2A
SCHEMBL7512580 0.82 BACE1 (0.65) BACE1ALDH1A1GRM2CTSDMEN1
SCHEMBL7518711 0.82 BACE1 (0.48) BACE1GRM2CTSD
SCHEMBL7518412 0.82 BACE1 (0.65) BACE1ALDH1A1GRM2CTSDMEN1
SCHEMBL12410201 0.81 BACE1 (0.53) BACE1ALDH1A1GRM2CTSDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2153832-B1 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2016-03-09 EP disclosed