SCHEMBL17572011

SCHEMBL17572011

O=NC(=O)c1ccc(Cl)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.56
CES1 P23141 3/20 0.56
TSHR P16473 2/20 0.54
ALOX15 P16050 1/20 0.54
CA1 P00915 2/20 0.52
CA2 P00918 2/20 0.52
GSK3B P49841 2/20 0.48
MAPK1 P28482 2/20 0.48
SRD5A2 P31213 1/20 0.48
L3MBTL1 Q9Y468 3/20 0.46
LMNA P02545 2/20 0.46
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
MAPT P10636 1/20 0.46
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19112012 0.87 HDAC8 (0.50) CES2CES1TSHRALOX15CA1
SCHEMBL26498861 0.79 HDAC3 (0.45) TSHRCA1CA2GSK3BL3MBTL1
SCHEMBL16729457 0.78 CES2 (0.54) CES2CES1TSHRALOX15CA1
SCHEMBL3822405 0.78 CES2 (0.54) CES2CES1TSHRALOX15CA1
SCHEMBL14879110 0.78 CES2 (0.61) CES2CES1TSHRALOX15CA1
SCHEMBL14997458 0.77 TSHR (0.63) CES2CES1TSHRALOX15CA1
SCHEMBL10363133 0.76 CES2 (0.52) CES2CES1TSHRALOX15CA1
SCHEMBL10363134 0.76 CES2 (0.52) CES2CES1TSHRALOX15CA1
SCHEMBL17733133 0.75 HDAC3 (0.47) TSHRCA1CA2MAPK1ALDH1A1
SCHEMBL4793883 0.75 CES2 (0.56) CES2CES1CA1CA2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016034671-A1 AMINOINDANE-, AMINOTETRAHYDRONAPHTHALENE- AND AMINOBENZOCYCLOBUTANE-DERIVED PRMT5-INHIBITORS CTXT PTY LTD (AU) 2016-03-10 WO disclosed