SCHEMBL17593153

SCHEMBL17593153

CCn1nc(-c2ccccc2)cc1C(=O)O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.56
POLB P06746 1/20 0.56
TDP1 Q9NUW8 2/20 0.49
ALDH1A1 P00352 3/20 0.48
HTT P42858 1/20 0.48
RAB9A P51151 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
MAPT P10636 1/20 0.46
PHGDH O43175 1/20 0.46
GABRP O00591 1/20 0.46
GABRD O14764 1/20 0.46
GABRA1 P14867 1/20 0.46
GABRB1 P18505 1/20 0.46
GABRG2 P18507 1/20 0.46
GABRB3 P28472 1/20 0.46
GABRA5 P31644 1/20 0.46
GABRA3 P34903 1/20 0.46
GABRA2 P47869 1/20 0.46
GABRB2 P47870 1/20 0.46
GABRA4 P48169 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28123448 0.88 SMN1; SMN2 (0.56) SMN1; SMN2POLBTDP1ALDH1A1MAPT
SCHEMBL596066 0.88 SMN1; SMN2 (0.53) SMN1; SMN2POLBTDP1ALDH1A1HTT
SCHEMBL28014537 0.86 HDAC6 (0.46) SMN1; SMN2POLBTDP1ALDH1A1RAB9A
SCHEMBL28013853 0.86 HDAC6 (0.60) SMN1; SMN2POLBTDP1MARS1HDAC6
SCHEMBL6335193 0.84 SMN1; SMN2 (0.79) SMN1; SMN2POLBTDP1ALDH1A1HTT
SCHEMBL4692309 0.84 PPARG (0.54) SMN1; SMN2POLBTDP1RAB9AMAPT
SCHEMBL14152218 0.84 PHGDH (0.46) SMN1; SMN2POLBTDP1ALDH1A1MAPT
SCHEMBL28013857 0.84 MARS1 (0.45) SMN1; SMN2POLBTDP1ALDH1A1MAPT
SCHEMBL4678362 0.83 HDAC6 (0.46) SMN1; SMN2POLBTDP1ALDH1A1MARS1
SCHEMBL27687138 0.83 SMN1; SMN2 (0.69) SMN1; SMN2POLBTDP1HTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016040449-A1 3-PHOSPHOGLYCERATE DEHYDROGENASE INHIBITORS AND USES THEREOF RAZE THERAPEUTICS, INC. (US) 2016-03-17 WO disclosed
CN-1230166-C Gyrase inhibitors and uses thereof VERTEX PHARMA (US) 2005-12-07 CN disclosed
CN-1400898-A Gyrase inhibitors and uses thereof VERTEX PHARMA (US) 2003-03-05 CN disclosed