SCHEMBL17594875

SCHEMBL17594875

CCc1cc(C(=O)OC(=O)C(F)(F)F)c(=O)[nH]c1-c1ccc(N2C[C@H]3CCC[C@@H](NC)[C@H]3C2)cc1

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 3/20 0.38
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
PARP1 P09874 1/20 0.31
PARP2 Q9UGN5 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17594910 0.89 CACNA1B (0.33) CACNA1BPDE3BPDE3APARP1PARP2
SCHEMBL17595147 0.89 CACNA1B (0.33) CACNA1BPDE3BPDE3APARP1PARP2
Trifluoroacetic Acid SCHEMBL14741141 0.88 CACNA1B (0.38) CACNA1BPDE3BPDE3APARP1PARP2
SCHEMBL16567996 0.87 CACNA1B (0.37) CACNA1BPDE3BPDE3APARP1PARP2
SCHEMBL14745237 0.85 CACNA1B (0.35) CACNA1BPARP1PARP2
SCHEMBL14745082 0.85 CACNA1B (0.35) CACNA1BPARP1PARP2
SCHEMBL14745545 0.85 PDE3B (0.32) CACNA1BPDE3BPDE3APARP1PARP2
SCHEMBL14741105 0.85 CACNA1B (0.31) CACNA1B
SCHEMBL17595205 0.83 PDE3B (0.35) PDE3BPDE3A
SCHEMBL16568463 0.82 PDE3B (0.34) PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016039936-A2 MONOCYCLIC SUBSTITUTED 2-PYRIDINONE ANTIBACTERIAL COMPOUNDS PTC THERAPEUTICS, INC. (US) 2016-03-17 WO claimed