SCHEMBL17598139

SCHEMBL17598139

CCc1c(-c2ccc3c(c2)NCCN3C)[nH]c(=O)c(C(=O)O)c1O

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 3/20 0.34
TLR8 Q9NR97 2/20 0.34
TLR9 Q9NR96 2/20 0.30
TNKS O95271 1/20 0.30
PARP1 P09874 1/20 0.30
TNKS2 Q9H2K2 1/20 0.30
MPL P40238 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL17597455 0.99 TLR8 (0.33) TLR7TLR8TLR9
SCHEMBL14741079 0.84 NOTUM (0.41) TLR7TLR8TNKSPARP1TNKS2
SCHEMBL14745370 0.83 NOTUM (0.44)
SCHEMBL14741280 0.82 PARP1 (0.39) TLR7TLR8TLR9TNKSPARP1
SCHEMBL17597633 0.81 JAK2 (0.36) TLR7TLR8
SCHEMBL17597124 0.81 PDE3B (0.42) PARP1
SCHEMBL17597194 0.79 MEN1 (0.31)
Hydrochloric Acid SCHEMBL17597730 0.78 MEN1 (0.33)
SCHEMBL14744809 0.78 ALDH1A1 (0.36) TLR7TLR8TLR9PARP1MPL
SCHEMBL14744987 0.77 ALDH1A1 (0.37) TLR7TLR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016039939-A1 BICYCLIC AND TRICYCLIC SUBSTITUTED 2-PYRIDINONE ANTIBACTERIAL COMPOUNDS PTC THERAPEUTICS, INC. (US) 2016-03-17 WO claimed
WO-2016039939-A1 BICYCLIC AND TRICYCLIC SUBSTITUTED 2-PYRIDINONE ANTIBACTERIAL COMPOUNDS PTC THERAPEUTICS, INC. (US) 2016-03-17 WO disclosed