SCHEMBL1759924

SCHEMBL1759924

CC(CCc1ccc(NC(=O)c2ccccc2)cc1)[C@H]1COC(N)=N1

nearest known ligand 0.68

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
KDM4E B2RXH2 1/20 0.44
MAPT P10636 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CCR2 P41597 1/20 0.42
TRPV1 Q8NER1 1/20 0.42
TAAR1 Q96RJ0 1/20 0.42
PPARA Q07869 1/20 0.42
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1760404 0.86 NPC1 (0.45) SMN1; SMN2
SCHEMBL1832205 0.82 TAAR1 (0.60) TAAR1
SCHEMBL1760021 0.78 TAAR1 (0.64) TAAR1
SCHEMBL1760023 0.78 TAAR1 (0.64) TAAR1
SCHEMBL1759920 0.78 TAAR1 (0.53) SMN1; SMN2TAAR1
SCHEMBL1774031 0.78 TAAR1 (0.53) SMN1; SMN2TAAR1
SCHEMBL1759746 0.76 TAAR1 (0.53) TAAR1
SCHEMBL1759747 0.76 TAAR1 (0.53) TAAR1
SCHEMBL502865 0.74
SCHEMBL1760187 0.74 TAAR1 (0.53) TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2499121-A1 OXAZOLINE DERIVATIVES FOR TREATMENT OF CNS DISORDERS. F. Hoffmann-La Roche AG (CH) 2012-09-19 EP disclosed
WO-2011057973-A1 OXAZOLINE DERIVATIVES FOR TREATMENT OF CNS DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2011-05-19 WO disclosed