SCHEMBL17599622

SCHEMBL17599622

CCC[C@](C)(COc1c(-c2cccc3c2CCC3=O)ccc(OC)c1OC)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 2/20 0.46
HPGD P15428 2/20 0.46
HDAC4 P56524 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
GAA P10253 2/20 0.35
PDE4D Q08499 1/20 0.34
S1PR1 P21453 1/20 0.34
BRAF P15056 1/20 0.34
MEN1 O00255 1/20 0.33
USP2 O75604 1/20 0.33
S100A4 P26447 1/20 0.33
KMT2A Q03164 1/20 0.33
TUBB4A P04350 1/20 0.33
TUBB P07437 1/20 0.33
TUBA3C P0DPH7 1/20 0.33
TUBA1B P68363 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17599590 1.00 ALDH1A1 (0.46) ALDH1A1KDM4EHPGDHDAC4HDAC2
SCHEMBL17599641 0.92 KDM4E (0.48) ALDH1A1KDM4EHPGDHDAC4HDAC2
SCHEMBL2593421 0.87 KDM4E (0.36) ALDH1A1KDM4EHPGDCNR1CNR2
SCHEMBL2591573 0.87 ALDH1A1 (0.51) ALDH1A1KDM4EHPGDHDAC4HDAC2
SCHEMBL17599591 0.83 KDM4E (0.47) ALDH1A1KDM4EHPGDHDAC4HDAC2
SCHEMBL17599642 0.83 KDM4E (0.47) ALDH1A1KDM4EHPGDHDAC4HDAC2
SCHEMBL2592149 0.82 ALDH1A1 (0.50) ALDH1A1KDM4EHPGDHDAC4HDAC2
SCHEMBL2588129 0.82 ALDH1A1 (0.50) ALDH1A1KDM4EHPGDHDAC4HDAC2
SCHEMBL14736959 0.82 ALDH1A1 (0.46) ALDH1A1KDM4EHPGDHDAC4HDAC2
SCHEMBL2592461 0.82 ALDH1A1 (0.46) ALDH1A1KDM4EHPGDHDAC4HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2563770-B1 BIARYL PHOSPHODIESTERASE INHIBITORS LEO PHARMA AS (DK) 2016-03-23 EP claimed