SCHEMBL17607252

SCHEMBL17607252

CN1CCC(Oc2ccc(NC(=O)c3ccc[nH]3)cn2)CC1

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAPK7 Q13164 1/20 0.60
DYRK1A Q13627 7/20 0.55
CLK2 P49760 5/20 0.55
CLK3 P49761 4/20 0.55
GSK3B P49841 3/20 0.54
NAMPT P43490 11/20 0.52
TDO2 P48775 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17607239 0.86 TMIGD3 (0.46) MAPK7DYRK1ACLK2CLK3NAMPT
SCHEMBL4506952 0.81 GSK3B (0.50) MAPK7DYRK1AGSK3BNAMPT
SCHEMBL20265901 0.76 MAPK7 (1.00) MAPK7
SCHEMBL22235838 0.72 DYRK1A (0.59) MAPK7DYRK1ACLK2CLK3GSK3B
SCHEMBL22236189 0.71 DYRK1A (0.59) MAPK7DYRK1ACLK2CLK3GSK3B
SCHEMBL22235982 0.71 DYRK1A (0.75) MAPK7DYRK1ACLK2CLK3GSK3B
SCHEMBL22235957 0.71 DYRK1A (0.59) MAPK7DYRK1ACLK2CLK3GSK3B
SCHEMBL17096486 0.71 DYRK1A (0.77) DYRK1ACLK2CLK3GSK3B
SCHEMBL22236116 0.71 DYRK1A (0.64) MAPK7DYRK1ACLK2CLK3GSK3B
SCHEMBL23449166 0.71 EHMT2 (0.56) MAPK7DYRK1ACLK2CLK3GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3194390-A1 PYRROLCARBOXAMIDE DERIVATIVES FOR THE INHBITION OF ERK5 Cancer Research Technology Ltd (GB) 2017-07-26 EP claimed
WO-2016042341-A1 PYRROLCARBOXAMIDE DERIVATIVES FOR THE INHBITION OF ERK5 CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2016-03-24 WO claimed