SCHEMBL17609342

SCHEMBL17609342

O=C1CCc2cc(C(=O)CN3CSC(=C4CCCCC4)C3)ccc2N1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 2/20 0.49
HTR1A P08908 2/20 0.42
HTR2A P28223 2/20 0.42
HTR7 P34969 2/20 0.42
DRD3 P35462 2/20 0.42
DRD4 P21917 1/20 0.42
CRBN Q96SW2 6/20 0.41
HDAC3 O15379 2/20 0.40
HDAC4 P56524 2/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC2 Q92769 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
HDAC9 Q9UKV0 2/20 0.40
DRD2 P14416 1/20 0.39
HTR2C P28335 1/20 0.39
HTR2B P41595 1/20 0.39
SMYD3 Q9H7B4 1/20 0.39
ALDH1A1 P00352 2/20 0.37
CYP2C9 P11712 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11255645 0.79 GRIN2B (0.57) GRIN2BHTR1AHTR2AHTR7DRD3
SCHEMBL17621231 0.76 GRIN2B (0.45) GRIN2BHTR1AHTR2AHTR7DRD3
SCHEMBL7344494 0.74 GRIN2B (0.57) GRIN2BHTR1AHTR2AHTR7DRD3
SCHEMBL5069516 0.74 GRIN2B (0.50) GRIN2BHTR1AHTR2AHTR7DRD3
Bromide SCHEMBL3843849 0.74 GRIN2B (0.49) GRIN2BHTR1AHTR2AHTR7DRD3
SCHEMBL8440778 0.73 GRIN2B (0.53) GRIN2BHTR1AHTR2AHTR7DRD3
Hydrochloric Acid SCHEMBL7349822 0.73 GRIN2B (0.55) GRIN2BHTR1AHTR2AHTR7DRD3
Hydrochloric Acid SCHEMBL10838416 0.73 GRIN2B (0.55) GRIN2BHTR1AHTR2AHTR7DRD3
SCHEMBL8439771 0.71 GRIN2B (0.52) GRIN2BHTR1AHTR2AHTR7DRD3
SCHEMBL2641171 0.70 CRBN (0.51) GRIN2BHTR1AHTR2AHTR7DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016044771-A1 HAT INHIBITORS AND METHODS FOR THEIR USE ABBVIE INC. (US) 2016-03-24 WO claimed