SCHEMBL8440778

SCHEMBL8440778

O=C1CCc2cc(C(=O)CN3CCC(CCC4CCCCC4)CC3)ccc2N1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 2/20 0.53
ACHE P22303 8/20 0.46
CRBN Q96SW2 3/20 0.46
HTR1A P08908 1/20 0.45
DRD4 P21917 1/20 0.45
HTR2A P28223 1/20 0.45
HTR7 P34969 1/20 0.45
DRD3 P35462 1/20 0.45
SMYD3 Q9H7B4 1/20 0.44
ALDH1A1 P00352 2/20 0.44
CRHBP P24387 1/20 0.44
CRHR2 Q13324 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KDM4E B2RXH2 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HTR4 Q13639 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8439771 0.96 GRIN2B (0.52) GRIN2BACHECRBNHTR1ADRD4
SCHEMBL8302305 0.90 GRIN2B (0.52) GRIN2BACHEHTR1AHTR2AHTR7
SCHEMBL7328182 0.86 GRIN2B (0.62) GRIN2BACHECRBNHTR1ADRD4
Hydrochloric Acid SCHEMBL11255645 0.85 GRIN2B (0.57) GRIN2BCRBNHTR1ADRD4HTR2A
SCHEMBL2237118 0.82 SMYD3 (0.51) GRIN2BCRBNHTR1ADRD4HTR2A
SCHEMBL7344494 0.81 GRIN2B (0.57) GRIN2BCRBNHTR1ADRD4HTR2A
SCHEMBL8543583 0.80 ACHE (0.60) GRIN2BACHE
Hydrochloric Acid SCHEMBL10838416 0.79 GRIN2B (0.55) GRIN2BCRBNHTR1ADRD4HTR2A
Hydrochloric Acid SCHEMBL7349822 0.79 GRIN2B (0.55) GRIN2BCRBNHTR1ADRD4HTR2A
SCHEMBL5470505 0.78 GRIN2B (0.53) GRIN2BCRBNHTR1ADRD4HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888340-A1 4-(BENZO-1,3-DIOXOLYL)-PYRROLIDINE-3-CARBOXYLIC ACID DERIVATIVES AS ENDOTHELIN ANTAGONISTS Abbott Laboratories (US) 1999-01-07 EP claimed
WO-1997030046-A1 4-(BENZO-1,3-DIOXOLYL)-PYRROLIDINE-3-CARBOXYLIC ACID DERIVATIVES AS ENDOTHELIN ANTAGONISTS ABBOTT LABORATORIES (US) 1997-08-21 WO claimed
EP-0848707-B1 4-(CYCLOALKYL)PIPERIDINES AND 4-(CYCLOALKYLALKYL)-PIPERIDINES DERIVATIVES, PREPARATION THEREOF AND THERAPEUTICAL APPLICATIONS THEREOF SYNTHELABO (FR) 1999-08-04 EP disclosed