SCHEMBL17612970

SCHEMBL17612970

COc1c(CN2C(C)CCC2C)cc(C(F)(F)F)cc1NC(=O)c1ccc(Cl)c(-n2cc(-c3cnn(C)c3C)n2C)c1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BRAF P15056 6/20 0.38
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP2C9 P11712 1/20 0.37
MAPT P10636 2/20 0.36
TP53 P04637 1/20 0.34
CYP2D6 P10635 1/20 0.34
RORC P51449 1/20 0.32
HTR2A P28223 3/20 0.32
HTR2C P28335 1/20 0.32
ABL1 P00519 1/20 0.32
NR2E1 Q9Y466 1/20 0.32
ACKR3 P25106 1/20 0.31
POLB P06746 1/20 0.31
MAPK14 Q16539 1/20 0.31
MAP3K20 Q9NYL2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17612974 0.89 BRAF (0.41) BRAFABL1
SCHEMBL12397281 0.87 ABL1 (0.40) BRAFCYP1A2CYP3A4CYP2C19CYP2C9
SCHEMBL13960393 0.79 BRAF (0.37) BRAFCYP1A2CYP3A4CYP2C19CYP2C9
SCHEMBL12397363 0.77 ABL1 (0.44) BRAFABL1
SCHEMBL12397372 0.77 ABL1 (0.42) BRAFABL1
SCHEMBL12397347 0.77 ABL1 (0.46) BRAFABL1
SCHEMBL12397355 0.77 ABL1 (0.46) BRAFABL1
SCHEMBL17612891 0.77 BRAF (0.42) BRAFCYP2C9MAPTABL1ACKR3
SCHEMBL12397291 0.76 ABL1 (0.51) ABL1
SCHEMBL12464981 0.76 ABL1 (0.40) BRAFABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2173734-B1 CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INT (DE) 2016-03-23 EP disclosed