SCHEMBL17612977

SCHEMBL17612977

COc1c(CN2CCC(O)CC2)cc(C(F)(F)F)cc1NC(=O)c1ccc(C)c(-n2cc(-c3cnn(C)c3C)[nH]2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 7/20 0.46
POLB P06746 1/20 0.38
PDCD1 Q15116 1/20 0.38
CD274 Q9NZQ7 1/20 0.38
KIT P10721 3/20 0.38
CSF1R P07333 2/20 0.38
CSK P41240 4/20 0.37
MAPK14 Q16539 4/20 0.37
DDR1 Q08345 1/20 0.37
MAP3K7 O43318 3/20 0.37
MAP4K2 Q12851 3/20 0.37
EPHA2 P29317 2/20 0.37
MAP3K20 Q9NYL2 2/20 0.37
ACKR3 P25106 1/20 0.37
BTK Q06187 2/20 0.36
HCK P08631 1/20 0.36
NR2C2 P49116 1/20 0.36
MAP4K4 O95819 1/20 0.36
ABL1 P00519 1/20 0.36
RAF1 P04049 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17612864 0.87 BRAF (0.43) BRAFPOLBACKR3ABL1
SCHEMBL12397429 0.87 ABL1 (0.48) BRAFABL1
SCHEMBL17612997 0.85 DDR2 (0.50) BRAFKITDDR1ABL1
SCHEMBL12397024 0.83 ABL1 (0.48) BRAFABL1
SCHEMBL12397363 0.82 ABL1 (0.44) BRAFABL1
SCHEMBL12397428 0.81 ABL1 (0.46) BRAFABL1
SCHEMBL12397437 0.80 ABL1 (0.49) BRAFABL1
SCHEMBL12397016 0.80 ABL1 (0.49) BRAFABL1
SCHEMBL12397439 0.80 ABL1 (0.55) ABL1
SCHEMBL12397431 0.79 ABL1 (0.51) BRAFABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2173734-B1 CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INT (DE) 2016-03-23 EP disclosed