SCHEMBL17614031

SCHEMBL17614031

CCOc1c(O)ccc(-c2cccc3c2CNC3=O)c1OCC(=O)OC1CCC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 12/20 0.35
ROCK1 Q13464 3/20 0.35
PLK4 O00444 2/20 0.35
ROCK2 O75116 2/20 0.35
NTRK1 P04629 2/20 0.35
MET P08581 2/20 0.35
ROS1 P08922 2/20 0.35
RPS6KB1 P23443 2/20 0.35
EPHA2 P29317 2/20 0.35
AXL P30530 2/20 0.35
FLT4 P35916 2/20 0.35
FLT3 P36888 2/20 0.35
FRK P42685 2/20 0.35
NTRK2 Q16620 2/20 0.35
TAOK1 Q7L7X3 2/20 0.35
HIPK4 Q8NE63 2/20 0.35
AURKB Q96GD4 2/20 0.35
SRPK1 Q96SB4 2/20 0.35
SRMS Q9H3Y6 2/20 0.35
ALK Q9UM73 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2591016 0.89 KDR (0.36) KDRROCK1PLK4ROCK2NTRK1
SCHEMBL2588770 0.87 KDR (0.36) KDRROCK1PLK4ROCK2NTRK1
SCHEMBL17613981 0.85 KDR (0.39) KDRROCK1PLK4ROCK2NTRK1
SCHEMBL17614021 0.85 PIK3CD (0.39) KDRROCK1PLK4ROCK2NTRK1
SCHEMBL2591886 0.84 KDR (0.38) KDRROCK1PLK4ROCK2NTRK1
SCHEMBL17613862 0.83 PIK3CD (0.35) KDRROCK1PLK4ROCK2NTRK1
SCHEMBL2589484 0.82 KDR (0.38) KDRROCK1PLK4ROCK2NTRK1
SCHEMBL17613865 0.82 ALDH1A1 (0.33) MAPTSMN1; SMN2ALDH1A1
SCHEMBL14737000 0.78 PIK3CD (0.34) KDRROCK1PLK4ROCK2NTRK1
SCHEMBL2591337 0.77 KDR (0.40) KDRROCK1PLK4ROCK2NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2563770-B1 BIARYL PHOSPHODIESTERASE INHIBITORS LEO PHARMA AS (DK) 2016-03-23 EP disclosed