SCHEMBL17620895

SCHEMBL17620895

COc1cccc(OC)c1CNC(=N)Nc1ccc2ccccc2n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.48
RAB9A P51151 6/20 0.48
CASP3 P42574 1/20 0.47
SENP7 Q9BQF6 1/20 0.47
SENP6 Q9GZR1 1/20 0.47
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
NOTUM Q6P988 1/20 0.46
NCF1 P14598 1/20 0.44
HTR1A P08908 4/20 0.41
NOD2 Q9HC29 1/20 0.41
ADORA2A P29274 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CNR2 P34972 1/20 0.40
DRD2 P14416 1/20 0.39
ADRA1A P35348 1/20 0.39
DRD3 P35462 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL2782911 0.94 NPC1 (0.49) NPC1RAB9ACASP3SENP7SENP6
SCHEMBL4629834 0.88 KMT2A (0.60) NPC1RAB9ACASP3SENP7SENP6
Acetic Acid SCHEMBL2779550 0.83 MEN1 (0.60) NPC1RAB9ACASP3SENP7SENP6
SCHEMBL2782719 0.81 KMT2A (0.49) NPC1RAB9AKMT2AMEN1SMN1; SMN2
SCHEMBL2779634 0.80 RXFP1 (0.40) NPC1RAB9AKMT2AMEN1SMN1; SMN2
SCHEMBL2780727 0.80 NOTUM (0.47) NPC1RAB9AKMT2AMEN1NOTUM
SCHEMBL2782180 0.80 ADORA3 (0.48) KMT2AADORA2ARXFP1ALDH1A1
SCHEMBL2777872 0.79 KDM4E (0.56) NPC1RAB9AKMT2AMEN1NOTUM
SCHEMBL2780656 0.79 NPC1 (0.52) NPC1RAB9AKMT2AMEN1SMN1; SMN2
SCHEMBL2779768 0.78 ADORA2A (0.44) NPC1RAB9AKMT2AMEN1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9296697-B2 Hetaryl-substituted guanidine compounds and use thereof as binding partners for 5-HT5-receptors ABBOTT LABORATORIES (US) 2016-03-29 US claimed