SCHEMBL17620899

SCHEMBL17620899

COc1ccccc1CN=C(N)Nc1ccc(-c2ccc(F)cc2)cn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK2 P49760 1/20 0.48
GSK3A P49840 1/20 0.48
GSK3B P49841 1/20 0.48
CDK9 P50750 1/20 0.48
CDK5 Q00535 1/20 0.48
DYRK1A Q13627 1/20 0.48
TAOK1 Q7L7X3 1/20 0.48
CLK4 Q9HAZ1 1/20 0.48
DYRK1B Q9Y463 1/20 0.48
ABCB1 P08183 2/20 0.42
GRIN2B Q13224 3/20 0.41
GRIN1 Q05586 2/20 0.41
ABCC1 P33527 1/20 0.41
ADRA2A P08913 3/20 0.40
ADRA2B P18089 3/20 0.40
ADRA2C P18825 3/20 0.40
KMT2A Q03164 1/20 0.40
GAA P10253 1/20 0.40
HTR7 P34969 1/20 0.40
ATM Q13315 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2781877 0.85 GSK3B (0.51) CLK2GSK3AGSK3BCDK9CDK5
SCHEMBL2781207 0.84 ABCB1 (0.42) ABCB1ABCC1KMT2AGAAWNT3A
SCHEMBL2780985 0.83 CLK2 (0.50) CLK2GSK3AGSK3BCDK9CDK5
SCHEMBL2781682 0.83 CLK2 (0.50) CLK2GSK3AGSK3BCDK9CDK5
SCHEMBL2780813 0.82 CLK2 (0.49) CLK2GSK3AGSK3BCDK9CDK5
SCHEMBL2781549 0.80 CLK4 (0.48) CLK2GSK3AGSK3BCDK9CDK5
SCHEMBL2779819 0.80 CLK2 (0.48) CLK2GSK3AGSK3BCDK9CDK5
SCHEMBL2781794 0.79 CLK4 (0.48) CLK2GSK3AGSK3BCDK9CDK5
SCHEMBL2782306 0.79 GRIN2B (0.54) CLK2GSK3AGSK3BCDK9CDK5
SCHEMBL17620898 0.77 KMT2A (0.48) ABCB1ABCC1KMT2AGAAATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9296697-B2 Hetaryl-substituted guanidine compounds and use thereof as binding partners for 5-HT5-receptors ABBOTT LABORATORIES (US) 2016-03-29 US claimed