SCHEMBL17620898

SCHEMBL17620898

COc1ccccc1CNC(=N)Nc1ccc(-c2ccc(F)cc2)cn1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.48
ROCK2 O75116 1/20 0.47
HTT P42858 1/20 0.46
ATM Q13315 1/20 0.46
GAA P10253 1/20 0.45
PLA2G1B P04054 1/20 0.45
ATG4B Q9Y4P1 1/20 0.45
ABCB1 P08183 2/20 0.43
MAPK1 P28482 2/20 0.42
POLB P06746 2/20 0.42
MEN1 O00255 1/20 0.42
TP53 P04637 3/20 0.42
ABCC1 P33527 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL2781206 0.95 HTT (0.49) KMT2AROCK2HTTGAAPLA2G1B
SCHEMBL2781937 0.93 HTT (0.53) KMT2AROCK2HTTATMGAA
SCHEMBL2782775 0.89 HTT (0.45) KMT2AROCK2HTTATMGAA
SCHEMBL17620892 0.88 ROCK2 (0.47) ROCK2ABCB1MAPK1ABCC1
Acetic Acid SCHEMBL2780720 0.85 HTT (0.48) KMT2AROCK2HTTGAAMAPK1
SCHEMBL2781874 0.85 KMT2A (0.46) KMT2AROCK2HTTGAAPLA2G1B
SCHEMBL2781226 0.84 MEN1 (0.51) KMT2AROCK2ATMGAAPOLB
SCHEMBL4629710 0.84 KMT2A (0.53) KMT2AROCK2ATMGAAMAPK1
Acetic Acid SCHEMBL2781275 0.83 ROCK2 (0.48) ROCK2GAAABCB1MAPK1ABCC1
SCHEMBL2780981 0.83 ATM (0.48) KMT2AROCK2HTTATMGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9296697-B2 Hetaryl-substituted guanidine compounds and use thereof as binding partners for 5-HT5-receptors ABBOTT LABORATORIES (US) 2016-03-29 US claimed