SCHEMBL17630083

SCHEMBL17630083

CC(C)C(=O)NCCCc1cc(C#N)ccc1-c1ccc(Br)cc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 1/20 0.42
TBXA2R P21731 1/20 0.38
CNR1 P21554 2/20 0.37
CNR2 P34972 1/20 0.37
MMP2 P08253 1/20 0.37
MMP3 P08254 1/20 0.37
MTNR1A P48039 3/20 0.36
MTNR1B P49286 3/20 0.36
PTGES O14684 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CTSK P43235 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17630196 0.81 GRIA1 (0.45) TBXA2R
SCHEMBL17630080 0.80 PDE2A (0.46) L3MBTL1
SCHEMBL17629919 0.79 KDM1A (0.37) CNR1
SCHEMBL17629879 0.79 KMT2A (0.48) CYP2D6CYP2C9CYP2C19KMT2ATBXA2R
SCHEMBL17629922 0.75 KDM1A (0.41) KMT2AMMP2MMP3
SCHEMBL17630064 0.74 PDE2A (0.46)
SCHEMBL17630007 0.73 HRH2 (0.36)
SCHEMBL17630076 0.72 HRH2 (0.35) L3MBTL1
SCHEMBL17629872 0.71 HSD17B10 (0.44) CYP2D6CYP2C9CYP2C19KMT2AMMP2
SCHEMBL17672870 0.70 CYP2D6 (0.39) CYP2D6CYP2C9CYP2C19KMT2AMTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016046782-A1 IMIDAZOLE BIARYL COMPOUNDS AS S-NITROSOGLUTATHIONE REDUCTASE INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2016-03-31 WO disclosed
WO-2016046782-A1 IMIDAZOLE BIARYL COMPOUNDS AS S-NITROSOGLUTATHIONE REDUCTASE INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2016-03-31 WO disclosed