SCHEMBL1763695

SCHEMBL1763695

C=CCC(=O)c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.61
CES1 P23141 2/20 0.55
CA1 P00915 2/20 0.53
CA2 P00918 2/20 0.53
TDP1 Q9NUW8 1/20 0.53
ALDH1A1 P00352 2/20 0.52
TSHR P16473 1/20 0.52
MAPK1 P28482 1/20 0.52
TGM2 P21980 1/20 0.51
KDM4E B2RXH2 1/20 0.50
LMNA P02545 1/20 0.50
HTT P42858 1/20 0.50
MAPT P10636 1/20 0.50
HSD11B1 P28845 1/20 0.49
CES2 O00748 1/20 0.49
SRD5A2 P31213 1/20 0.49
MMP8 P22894 1/20 0.48
PKM P14618 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2554642 0.84 GSK3B (0.62) GSK3BCES1CA1CA2TDP1
SCHEMBL5099884 0.79 CES1 (0.61) GSK3BCES1CA1CA2TDP1
SCHEMBL8024787 0.79 GSK3B (0.67) GSK3BCES1CA1CA2TDP1
SCHEMBL27694666 0.79 TSHR (0.49) GSK3BCES1CA1CA2TDP1
SCHEMBL2298238 0.79 MAPT (0.54) GSK3BCES1CA1CA2TDP1
SCHEMBL240086 0.79 GSK3B (0.71) GSK3BCES1CA1CA2TDP1
SCHEMBL11510574 0.79 GSK3B (0.71) GSK3BCES1CA1CA2TDP1
SCHEMBL28552870 0.78 CES1 (0.46) GSK3BCES1CA1CA2TDP1
SCHEMBL21782374 0.78 GSK3B (0.56) GSK3BCES1CA1CA2TDP1
SCHEMBL28552872 0.78 CES1 (0.46) GSK3BCES1CA1CA2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0269041-B1 FUNGICIDAL CYCLOHEXYLAMINES BASF Aktiengesellschaft (DE) 1991-04-10 EP claimed
US-4751304-A Process for preparing 5,6-dialkoxy-4-alkyl-2(1H)-quinazolinones ORTHO PHARMACEUTICAL CORPORATION (US) 1988-06-14 US claimed
EP-0177256-A2 Process for preparing 5,6-dialkoxy-4-alkyl-2(1h)-quinazolinones ORTHO PHARMACEUTICAL CORPORATION (US) 1986-04-09 EP claimed
JP-6092912-A None JP disclosed
CN-115710281-B Isoxazolo [5,4-b ] pyridine FLT3 inhibitor and preparation method and application thereof 南京中医药大学 2024-05-17 CN disclosed
CN-102105435-B 5-isopropyl-3-aminomethyl-2-methyl-1-amino-cyclohexane (carvone diamine), and method for the production thereof BASF SE 2014-07-23 CN disclosed
US-8586794-B2 5-isopropyl-3-aminomethyl-2-methyl-1-amino-cyclohexane (carvone diamine), and method for the production thereof BASF SE (DE) 2013-11-19 US disclosed
CN-102105434-A 3-aminomethyl-1-cyclohexylamine, and method for the production thereof BASF SE 2011-06-22 CN disclosed
CN-102105435-A 5-isopropyl-3-aminomethyl-2-methyl-1-amino-cyclohexane (carvone diamine), and method for the production thereof BASF SE 2011-06-22 CN disclosed
US-20110124918-A1 5-ISOPROPYL-3-AMINOMETHYL-2-METHYL-1-AMINO-CYCLOHEXANE (CARVONE DIAMINE), AND METHOD FOR THE PRODUCTION THEREOF BASF SE (DE) 2011-05-26 US disclosed
US-20110124919-A1 3-AMINOMETHYL-1-CYCLOHEXYLAMINE, AND METHOD FOR THE PRODUCTION THEREOF BASF SE (DE) 2011-05-26 US disclosed
US-5336749-A Alicyclic diamines, alicyclic diisocyanates and polyisocyanato-isocyanurates and method for the preparation thereof MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1994-08-09 US disclosed
JP-H0692912-A PRODUCTION OF DIAMINES MITSUI TOATSU CHEM INC 1994-04-05 JP disclosed
EP-0394058-B1 ALICYCLIC DIAMINES, ALICYCLIC DIISOCYANATES AND POLYISOCYANATO-ISOCYANURATES AND METHOD FOR THE PREPARATION THEREOF MITSUI TOATSU CHEMICALS, Inc. (JP) 1993-08-25 EP disclosed
US-5210286-A Hydrogenation of corresponding aromatic compound, reaction with phosgene MITSUI TOATSU CHEMICALS, INC. (JP) 1993-05-11 US disclosed
US-5126426-A Catalytic hydrogenation of aromatic diamine MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1992-06-30 US disclosed
EP-0394058-A1 Alicyclic diamines, alicyclic diisocyanates and polyisocyanato-isocyanurates and method for the preparation thereof MITSUI TOATSU CHEMICALS, Inc. (JP) 1990-10-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110124919-A1 3-AMINOMETHYL-1-CYCLOHEXYLAMINE, AND METHOD FOR THE PRODUCTION THEREOF PNMT, CBR3, ALKBH3 GSK3B 4271/4885CES1 2183/4885CA1 1518/4885
US-20110124918-A1 5-ISOPROPYL-3-AMINOMETHYL-2-METHYL-1-AMINO-CYCLOHEXANE (CARVONE DIAMINE), AND METHOD FOR THE PRODUCTION THEREOF CARM1, PNMT, CPNE4 GSK3B 4791/4885CES1 3416/4885CA1 987/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.