SCHEMBL176377

SCHEMBL176377

CN[C@@H](C)C(N)[C@@H](C(=O)N1CCC[C@H]1C(=O)Nc1cc2c(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)ncnc2cc1OC)C(C)(C)C

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EGFR P00533 17/20 0.61
ERBB2 P04626 5/20 0.59
ERBB4 Q15303 3/20 0.59
JAK3 P52333 2/20 0.54
GAK O14976 1/20 0.53
CYP3A4 P08684 3/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15050091 0.88 CYP3A4 (0.65) EGFRERBB2ERBB4JAK3GAK
SCHEMBL15050088 0.88 CYP3A4 (0.65) EGFRERBB2ERBB4JAK3GAK
Hydrochloric Acid SCHEMBL15050483 0.88 CYP3A4 (0.65) EGFRERBB2ERBB4JAK3GAK
Hydrochloric Acid SCHEMBL15050486 0.88 CYP3A4 (0.65) EGFRERBB2ERBB4JAK3GAK
SCHEMBL178188 0.84 CYP3A4 (0.58) EGFRERBB2CYP3A4
Hydrochloric Acid SCHEMBL176203 0.84 CYP3A4 (0.56) EGFRERBB2CYP3A4
SCHEMBL176198 0.83 CYP3A4 (0.54) EGFRERBB2ERBB4JAK3GAK
Hydrochloric Acid SCHEMBL176332 0.83 CYP3A4 (0.55) EGFRERBB2CYP3A4
Hydrochloric Acid SCHEMBL176298 0.82 EGFR (0.60) EGFRERBB2CYP3A4
Hydrochloric Acid SCHEMBL176888 0.81 EGFR (0.70) EGFRERBB2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611797-A2 QUINOLINE OR QUINAZOLINE DERIVATIVES WITH APOPTOSIS INDUCING ACTIVITY ON CELLS Hanmi Science Co., Ltd. (KR) 2013-07-10 EP disclosed
WO-2012030160-A2 QUINOLINE OR QUINAZOLINE DERIVATIVES WITH APOPTOSIS INDUCING ACTIVITY ON CELLS HANMI HOLDINGS CO., LTD. (KR) 2012-03-08 WO disclosed