SCHEMBL176198

SCHEMBL176198

CN[C@@H](C)C(N)[C@@H](C(=O)N1CCC[C@H]1C(=O)Nc1cc2c(Nc3ccc(N4CCN(CC5CC5)CC4)c(Cl)c3)ncnc2cc1OC)C(C)(C)C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.54
CYP2C9 P11712 2/20 0.49
CYP2C19 P33261 1/20 0.49
XIAP P98170 1/20 0.49
EGFR P00533 12/20 0.44
ERBB2 P04626 8/20 0.44
ERBB4 Q15303 5/20 0.44
LCK P06239 2/20 0.44
SRC P12931 2/20 0.44
GAK O14976 1/20 0.44
RIPK2 O43353 1/20 0.44
NR1I2 O75469 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
CHRM1 P11229 1/20 0.44
DRD2 P14416 1/20 0.44
ADRA2C P18825 1/20 0.44
SLC6A2 P23975 1/20 0.44
MC3R P41968 1/20 0.44
JAK3 P52333 1/20 0.44
SLC6A3 Q01959 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15050302 0.88 CYP3A4 (0.70) CYP3A4CYP2C9CYP2C19XIAPEGFR
SCHEMBL15050305 0.88 CYP3A4 (0.70) CYP3A4CYP2C9CYP2C19XIAPEGFR
Hydrochloric Acid SCHEMBL176332 0.84 CYP3A4 (0.55) CYP3A4CYP2C9CYP2C19XIAPEGFR
Hydrochloric Acid SCHEMBL176203 0.83 CYP3A4 (0.56) CYP3A4CYP2C9CYP2C19XIAPEGFR
SCHEMBL176377 0.83 EGFR (0.61) CYP3A4EGFRERBB2ERBB4GAK
SCHEMBL176991 0.83 EGFR (0.56) CYP3A4CYP2C9CYP2C19XIAPEGFR
SCHEMBL18334937 0.82 CYP3A4 (0.69) CYP3A4CYP2C9CYP2C19XIAPEGFR
SCHEMBL15075582 0.82 CYP3A4 (0.69) CYP3A4CYP2C9CYP2C19XIAPEGFR
SCHEMBL18334959 0.82 CYP3A4 (0.67) CYP3A4CYP2C9CYP2C19XIAPEGFR
SCHEMBL15075578 0.82 CYP3A4 (0.67) CYP3A4CYP2C9CYP2C19XIAPEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611797-A2 QUINOLINE OR QUINAZOLINE DERIVATIVES WITH APOPTOSIS INDUCING ACTIVITY ON CELLS Hanmi Science Co., Ltd. (KR) 2013-07-10 EP disclosed
WO-2012030160-A2 QUINOLINE OR QUINAZOLINE DERIVATIVES WITH APOPTOSIS INDUCING ACTIVITY ON CELLS HANMI HOLDINGS CO., LTD. (KR) 2012-03-08 WO disclosed