SCHEMBL176441

SCHEMBL176441

C[C@H](NC(=O)c1nn(C2CCCCC2)c2c1CCCCC2Cc1cccc(Cl)c1)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 5/20 0.54
CNR1 P21554 3/20 0.43
MAPK1 P28482 3/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
PTGER4 P35408 2/20 0.41
TRPV4 Q9HBA0 1/20 0.40
GPR139 Q6DWJ6 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ATM Q13315 1/20 0.37
NTSR1 P30989 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL176767 1.00 CNR2 (0.54) CNR2CNR1MAPK1ALDH1A1LMNA
SCHEMBL176628 0.92 MAPK1 (0.45) CNR2CNR1MAPK1ALDH1A1LMNA
SCHEMBL176606 0.92 MAPK1 (0.45) CNR2CNR1MAPK1ALDH1A1LMNA
SCHEMBL176620 0.91 CNR2 (0.48) CNR2CNR1MAPK1ALDH1A1LMNA
SCHEMBL176638 0.91 CNR2 (0.48) CNR2CNR1MAPK1ALDH1A1LMNA
SCHEMBL176782 0.87 MAPK1 (0.45) CNR2CNR1MAPK1ALDH1A1LMNA
SCHEMBL300678 0.87 CNR2 (0.48) CNR2MAPK1PTGER4TRPV4
SCHEMBL3466374 0.85 CNR2 (0.46) CNR2CNR1ALDH1A1
SCHEMBL176823 0.85 CNR2 (0.44) CNR2CNR1ALDH1A1MEN1KMT2A
SCHEMBL176650 0.84 EPHX2 (0.45) CNR2CNR1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937259-B1 HEXAHYDRO-CYCLOHEPTAPYRAZOLE CANNABINOID MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2011-11-23 EP disclosed