Formic Acid

Formic Acid

SCHEMBL1765337

O=C1CN(C(=O)c2cc(-c3cccc(OCCCN4CCC4)c3)n(-c3cccc(Cl)c3)n2)CN1.O=CO

nearest known ligand 0.45

Full drug profile on Sugi Atlas →

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCKAR P32238 1/20 0.45
HRH3 Q9Y5N1 8/20 0.41
AVPR1B P47901 3/20 0.39
PTGS2 P35354 2/20 0.39
PTGS1 P23219 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
SLC5A1 P13866 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Formic Acid SCHEMBL1765453 0.99 CCKAR (0.45) CCKARHRH3AVPR1B
SCHEMBL12597312 0.97 CCKAR (0.48) CCKARHRH3AVPR1BPTGS2PTGS1
SCHEMBL12597289 0.96 CCKAR (0.48) CCKARHRH3AVPR1BPTGS2
Formic Acid SCHEMBL1765088 0.94 CCKAR (0.46) CCKARHRH3AVPR1BPTGS2PTGS1
SCHEMBL12597317 0.91 CCKAR (0.48) CCKARHRH3AVPR1BPTGS2PTGS1
SCHEMBL12597299 0.91 PTGS2 (0.48) CCKARAVPR1BPTGS2KDM4E
Formic Acid SCHEMBL1764889 0.90 KDM4E (0.48) CCKARPTGS2KDM4EALDH1A1
Formic Acid SCHEMBL1764985 0.90 CCKAR (0.46) CCKARPTGS2PTGS1SLC5A1
Formic Acid SCHEMBL1765477 0.88 CCKAR (0.46) CCKARPTGS2PTGS1KDM4ESLC5A1
Formic Acid SCHEMBL1765040 0.88 CCKAR (0.46) CCKARSLC5A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8399682-B2 Substituted (pyrazolylcarbonyl)imidazolidinones and their use AICURIS GMBH & CO. KG (DE) 2013-03-19 US disclosed
US-20110124618-A1 SUBSTITUTED (PYRAZOLYLCARBONYL)IMIDAZOLIDINONES AND THEIR USE AICURIS GMBH & CO. KG (DE) 2011-05-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110124618-A1 SUBSTITUTED (PYRAZOLYLCARBONYL)IMIDAZOLIDINONES AND THEIR USE TPMT, PAICS, THPO CCKAR 4827/4885HRH3 744/4885AVPR1B 2782/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.