SCHEMBL17656285

SCHEMBL17656285

COC(=O)c1ccc(-c2ccc(C(=O)OC)cc2I)c(C)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 1/20 0.48
HCRTR2 O43614 1/20 0.48
CA1 P00915 3/20 0.47
CA2 P00918 3/20 0.47
CA12 O43570 2/20 0.47
CA7 P43166 2/20 0.47
CA9 Q16790 2/20 0.47
CA14 Q9ULX7 2/20 0.47
XDH P47989 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
PTPRC P08575 1/20 0.45
SLC2A1 P11166 1/20 0.44
MAPT P10636 4/20 0.44
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 2/20 0.44
HPGD P15428 2/20 0.44
HSD17B10 Q99714 2/20 0.44
GAA P10253 2/20 0.44
GLA P06280 1/20 0.44
CASP1 P29466 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL204112 0.91 CA1 (0.55) HCRTR1HCRTR2CA1CA2CA12
SCHEMBL16937873 0.89 TDP1 (0.57) CA1CA2CA12CA7CA9
SCHEMBL14950619 0.86 TDP1 (0.53) CA1CA2CA12CA7CA9
SCHEMBL14950616 0.86 TDP1 (0.53) CA1CA2CA12CA7CA9
SCHEMBL204113 0.85 KDM4E (0.53) HCRTR1HCRTR2CA1CA2CA12
SCHEMBL28268790 0.83 KDM4E (0.54) CA1CA2CA12CA7CA9
SCHEMBL1232173 0.82 TDP1 (0.53) HCRTR1HCRTR2CA1CA2CA12
SCHEMBL30010685 0.82 TDP1 (0.53) HCRTR1HCRTR2CA1CA2CA12
SCHEMBL1459771 0.82 TDP1 (0.53) HCRTR1HCRTR2CA1CA2CA12
SCHEMBL1529069 0.82 NOTUM (0.43) HCRTR1HCRTR2CA1CA2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3002281-B1 ANTIVIRAL COMPOUNDS GILEAD PHARMASSET LLC (US) 2017-09-13 EP disclosed
EP-3002281-A1 ANTIVIRAL COMPOUNDS Gilead Pharmasset LLC (US) 2016-04-06 EP disclosed