SCHEMBL17656300

SCHEMBL17656300

CC(C)(C)OC(=O)N1[C@@H]2CC[C@@H](C2)[C@H]1C(=O)OCC(=O)c1ccc2c(c1)COCc1cc(C(=O)CO)ccc1-2

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PREP P48147 4/20 0.41
CHRM2 P08172 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
ALDH1A1 P00352 3/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32
PDE4A P27815 2/20 0.32
PDE4B Q07343 2/20 0.32
PDE4C Q08493 2/20 0.32
PDE4D Q08499 2/20 0.32
HSD11B1 P28845 1/20 0.32
HTT P42858 1/20 0.32
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15368133 0.92 PREP (0.42) PREPCHRM2CHRM1CHRM3ALDH1A1
SCHEMBL9977159 0.92 PREP (0.42) PREPCHRM2CHRM1CHRM3ALDH1A1
SCHEMBL2708422 0.88 PREP (0.41) PREPALDH1A1MEN1KMT2ANPC1
SCHEMBL202883 0.88 PREP (0.41) PREPALDH1A1MEN1KMT2ANPC1
SCHEMBL18462482 0.88 PREP (0.41) PREPALDH1A1MEN1KMT2ANPC1
SCHEMBL19339404 0.87 PREP (0.36) PREPCHRM2CHRM1CHRM3ALDH1A1
SCHEMBL16891276 0.82 PREP (0.43) PREPCHRM2CHRM1CHRM3ALDH1A1
SCHEMBL17066298 0.82 PREP (0.50) PREPCHRM2CHRM1CHRM3ALDH1A1
SCHEMBL2709941 0.81 PREP (0.42) PREPALDH1A1MEN1KMT2ANPC1
SCHEMBL16001579 0.81 PREP (0.42) PREPALDH1A1MEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3002281-A1 ANTIVIRAL COMPOUNDS Gilead Pharmasset LLC (US) 2016-04-06 EP disclosed