SCHEMBL17664609

SCHEMBL17664609

CCNC(=O)c1nc(C(C)(C)C)no1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.40
KDM4E B2RXH2 1/20 0.40
HDAC4 P56524 2/20 0.39
HDAC6 Q9UBN7 2/20 0.39
PIK3CG P48736 1/20 0.39
BTK Q06187 9/20 0.38
HPGD P15428 2/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
LCK P06239 1/20 0.35
HDAC1 Q13547 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12410860 0.83 GAA (0.56) GAAKDM4EPIK3CGBTKSMN1; SMN2
SCHEMBL17660272 0.83 RAB9A (0.43) GAAKDM4EHDAC4PIK3CGBTK
SCHEMBL12321703 0.81 PIK3CG (0.41) GAAKDM4EHDAC4HDAC6PIK3CG
SCHEMBL12410863 0.81 PIK3CG (0.41) GAAKDM4EHDAC6PIK3CGBTK
SCHEMBL6119983 0.77 GAA (0.39) GAAKDM4EHDAC4HDAC6HPGD
SCHEMBL15221457 0.77 PIK3CG (0.39) GAAKDM4EHDAC4PIK3CGBTK
SCHEMBL12410869 0.77 KDM4E (0.43) GAAKDM4EPIK3CGBTKLCK
SCHEMBL4492502 0.75 KLKB1 (0.39) GAAKDM4EHDAC4HDAC6HPGD
SCHEMBL15662749 0.74 PIK3CG (0.41) GAAKDM4EPIK3CG
SCHEMBL17645642 0.74 PIK3CG (0.41) GAAKDM4EPIK3CGBTKTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240207267-A1 (R)-Glutarimide CRBN Ligands and Methods of Use BEIGENE SWITZERLAND GMBH (CH) 2024-06-27 US disclosed
US-10266528-B2 2-oxo-imidazopyridines as reversible BTK inhibitors and uses thereof MERCK PATENT GMBH (DE) 2019-04-23 US disclosed
WO-2018035080-A1 2-OXO-IMIDAZOPYRIDINES AS REVERSIBLE BTK INHIBITORS AND USES THEREOF MERCK PATENT GMBH (DE) 2018-02-22 WO disclosed
US-20180051024-A1 2-OXO-IMIDAZOPYRIDINES AS REVERSIBLE BTK INHIBITORS AND USES THEREOF MERCK PATENT GMBH (DE) 2018-02-22 US disclosed
US-20160096834-A1 HETEROARYL COMPOUNDS AS BTK INHIBITORS AND USES THEREOF MERCK PATENT GMBH (DE) 2016-04-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10266528-B2 2-oxo-imidazopyridines as reversible BTK inhibitors and uses thereof BTK, SYK, LCK GAA 3416/4885KDM4E 783/4885HDAC4 1057/4885
US-20160096834-A1 HETEROARYL COMPOUNDS AS BTK INHIBITORS AND USES THEREOF BTK, SYK, LYN GAA 2202/4885KDM4E 935/4885HDAC4 1733/4885
US-20240207267-A1 (R)-Glutarimide CRBN Ligands and Methods of Use CRBN, CDR2, CRKL GAA 1405/4885KDM4E 1286/4885HDAC4 2272/4885
US-20180051024-A1 2-OXO-IMIDAZOPYRIDINES AS REVERSIBLE BTK INHIBITORS AND USES THEREOF BTK, SYK, LCK GAA 3416/4885KDM4E 783/4885HDAC4 1057/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.