SCHEMBL17667296

SCHEMBL17667296

CC(C)(C)N(C(=O)O)[C@@H]1CCCN(c2nc(Cl)nc3cccnc23)C1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 2/20 0.40
RORC P51449 3/20 0.36
HRH4 Q9H3N8 1/20 0.35
JAK2 O60674 1/20 0.35
JAK3 P52333 1/20 0.35
CNR2 P34972 3/20 0.35
PDE10A Q9Y233 2/20 0.34
CCNE2 O96020 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
TLR7 Q9NYK1 1/20 0.34
KMT2A Q03164 1/20 0.34
TRPV1 Q8NER1 1/20 0.34
PIK3CD O00329 1/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CG P48736 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17667297 1.00 PRKDC (0.40) PRKDCRORCHRH4JAK2JAK3
SCHEMBL17628237 0.81 OPRM1 (0.46) PRKDCHRH4JAK2JAK3PDE10A
SCHEMBL17667319 0.81 JAK2 (0.39) RORCHRH4JAK2JAK3CNR2
SCHEMBL17628165 0.77 JAK2 (0.39) RORCHRH4JAK2JAK3PDE10A
SCHEMBL17628378 0.77 PRKDC (0.44) PRKDCCNR2PDE10AKMT2APIK3CA
SCHEMBL15929081 0.77 EIF2AK4 (0.42) HRH4TRPV1
SCHEMBL17667317 0.77 PDE10A (0.56) PRKDCJAK2JAK3CNR2PDE10A
SCHEMBL17628072 0.77 CNR2 (0.47) PRKDCCNR2PDE10AKMT2APIK3CD
SCHEMBL17628070 0.77 CNR2 (0.47) PRKDCCNR2PDE10AKMT2APIK3CD
SCHEMBL17667365 0.75 HRH4 (0.36) PRKDCHRH4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3006439-A1 BICYCLIC DERIVATIVE CONTAINING PYRIMIDINE RING, AND PREPARATION METHOD THEREFOR Yuhan Corporation (KR) 2016-04-13 EP disclosed