SCHEMBL17667883

SCHEMBL17667883

Nc1nnc(-c2cc(C[C@H](N)C(=O)O)cc(OC(F)(F)F)c2)c(-c2ccccc2)n1

nearest known ligand 0.48

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 14/20 0.48
ADORA1 P30542 14/20 0.48
ADORA2B P29275 2/20 0.42
TPH1 P17752 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2321936 0.79 ADORA2A (0.57) ADORA2AADORA1ADORA2B
SCHEMBL2326085 0.77 ADORA2A (0.57) ADORA2AADORA1ADORA2B
SCHEMBL2320490 0.76 ADORA2A (0.65) ADORA2AADORA1ADORA2B
SCHEMBL869894 0.72 TPH1 (0.61) TPH1
SCHEMBL869893 0.72 TPH1 (0.61) TPH1
SCHEMBL793094 0.71 SLC7A5 (0.57)
SCHEMBL793095 0.71 SLC7A5 (0.57)
SCHEMBL1802025 0.68 PTPN1 (0.78) TPH1
SCHEMBL18256435 0.68 PTPN1 (0.78) TPH1
SCHEMBL1802026 0.68 PTPN1 (0.78) TPH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2531492-B1 1,2,4-TRIAZINE-4-AMINE DERIVATIVES HEPTARES THERAPEUTICS LTD (GB) 2016-04-13 EP disclosed