SCHEMBL17674201

SCHEMBL17674201

O=C(O)n1c(-c2ncco2)cc2cc(F)ccc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 4/20 0.48
NTRK3 Q16288 3/20 0.48
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
HCRTR1 O43613 2/20 0.37
HCRTR2 O43614 2/20 0.37
CTSA P10619 4/20 0.37
ADRA1A P35348 2/20 0.34
TUBB4A P04350 1/20 0.34
TUBB P07437 1/20 0.34
TUBA3C P0DPH7 1/20 0.34
TUBA1B P68363 1/20 0.34
TUBA4A P68366 1/20 0.34
TUBB4B P68371 1/20 0.34
TUBB3 Q13509 1/20 0.34
TUBB2A Q13885 1/20 0.34
TUBB8 Q3ZCM7 1/20 0.34
TUBA3E Q6PEY2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17674395 0.83 NTRK3 (0.52) NTRK1NTRK3KDM4EALDH1A1HPGD
SCHEMBL17674391 0.81 NTRK1 (0.60) NTRK1NTRK3CTSA
SCHEMBL17674288 0.78 NTRK1 (0.59) NTRK1NTRK3HCRTR1HCRTR2CTSA
SCHEMBL17674286 0.78 NTRK1 (0.48) NTRK1NTRK3KDM4EALDH1A1HPGD
SCHEMBL17674258 0.75 KDM4E (0.46) NTRK1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL17674413 0.73 KDM4E (0.43) NTRK1NTRK3KDM4EALDH1A1HPGD
SCHEMBL27830572 0.72 ACLY (0.47) NTRK1
SCHEMBL17680336 0.71 NTRK1 (0.52) NTRK1NTRK3ALDH1A1
SCHEMBL3309831 0.70 GRM2 (0.38) NTRK1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL31196173 0.69 AOC3 (0.47) ALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016054807-A1 TrkA KINASE INHIBITORS, COMPOSITIONS AND METHODS THEREOF MERCK SHARP & DOHME CORP. (US) 2016-04-14 WO disclosed