SCHEMBL17675232

SCHEMBL17675232

C=CC(=O)Nc1cc2c(Oc3ccc(C(=O)Nc4ccccn4)cc3)ccnc2cc1OCCCn1cccc1

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BTK Q06187 17/20 0.64
EGFR P00533 15/20 0.64
TEC P42680 3/20 0.57
TXK P42681 3/20 0.57
BLK P51451 3/20 0.57
BMX P51813 3/20 0.57
ERBB4 Q15303 3/20 0.57
ERBB2 P04626 2/20 0.52
JAK3 P52333 2/20 0.52
ITK Q08881 1/20 0.52
CHRNB2 P17787 1/20 0.44
CHRNB4 P30926 1/20 0.44
CHRNA3 P32297 1/20 0.44
CHRNA4 P43681 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17675246 0.90 BTK (0.68) BTKEGFRTECTXKBLK
SCHEMBL17675231 0.90 BTK (0.70) BTKEGFRTECTXKBLK
SCHEMBL17675376 0.89 BTK (0.69) BTKEGFRTECTXKBLK
SCHEMBL17675526 0.88 BTK (0.79) BTKEGFRTECTXKBLK
SCHEMBL17675611 0.87 BTK (0.68) BTKEGFRTECTXKBLK
SCHEMBL17675620 0.87 BTK (0.64) BTKEGFRTECTXKBLK
SCHEMBL17675359 0.87 BTK (0.67) BTKEGFRTECTXKBLK
SCHEMBL17675333 0.87 BTK (0.81) BTKEGFRTECTXKBLK
SCHEMBL17675198 0.86 BTK (0.65) BTKEGFRTECTXKBLK
SCHEMBL17675259 0.86 BTK (0.73) BTKEGFRTECTXKBLK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016055982-A1 QUINOLINE AND QUINAZOLINE COMPOUNDS ACERTA PHARMA B.V. (NL) 2016-04-14 WO disclosed