SCHEMBL17675288

SCHEMBL17675288

O=C(Nc1ccc(C(F)(F)F)cn1)c1ccc(Oc2ccnc3ccc([N+](=O)[O-])cc23)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.48
RAB9A P51151 2/20 0.48
NPC1 O15118 1/20 0.48
ALDH1A1 P00352 1/20 0.48
LMNA P02545 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
BTK Q06187 6/20 0.48
EGFR P00533 5/20 0.48
KDR P35968 4/20 0.47
PDGFRA P16234 2/20 0.47
PTGS1 P23219 1/20 0.47
HTT P42858 1/20 0.46
NPSR1 Q6W5P4 1/20 0.45
USP2 O75604 1/20 0.45
KMT2A Q03164 1/20 0.45
IDO1 P14902 1/20 0.45
MET P08581 2/20 0.45
ERBB2 P04626 1/20 0.44
TEC P42680 1/20 0.44
TXK P42681 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17675515 0.90 BTK (0.49) MAPTBTKEGFRKDRPDGFRA
SCHEMBL17675318 0.84 BTK (0.66) MAPTRAB9ANPC1ALDH1A1LMNA
SCHEMBL17675295 0.83 KDR (0.48) MAPTBTKEGFRKDRPDGFRA
SCHEMBL17675511 0.82 KMT2A (0.55) MAPTRAB9ANPC1ALDH1A1LMNA
SCHEMBL17675493 0.80 BTK (0.68) MAPTRAB9ANPC1SMN1; SMN2BTK
SCHEMBL17675293 0.78 EGFR (0.49) MAPTRAB9ABTKEGFRKDR
SCHEMBL17675471 0.76 BTK (0.52) RAB9ANPC1ALDH1A1SMN1; SMN2BTK
SCHEMBL17675216 0.75 BTK (0.54) MAPTBTKEGFRKDRPTGS1
SCHEMBL30354762 0.75 MAPT (0.77) MAPTRAB9ANPC1ALDH1A1LMNA
SCHEMBL13428702 0.75 MAPT (0.77) MAPTRAB9ANPC1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016055982-A1 QUINOLINE AND QUINAZOLINE COMPOUNDS ACERTA PHARMA B.V. (NL) 2016-04-14 WO disclosed