SCHEMBL17675397

SCHEMBL17675397

CC#CC(=O)Nc1cc2c(Nc3ccc(C(=O)Nc4ccccn4)cc3)ncnc2cc1OC

nearest known ligand 0.70

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BTK Q06187 5/20 0.70
AURKB Q96GD4 4/20 0.59
AURKA O14965 2/20 0.59
EGFR P00533 5/20 0.58
KDR P35968 8/20 0.56
ERBB4 Q15303 2/20 0.55
ERBB2 P04626 1/20 0.55
MAPK14 Q16539 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17675602 0.89 BTK (0.76) BTKAURKBAURKAEGFRKDR
SCHEMBL17675257 0.87 EGFR (0.72) BTKAURKBAURKAEGFRKDR
SCHEMBL17675217 0.86 KDR (0.63) BTKAURKBAURKAEGFRKDR
SCHEMBL17683840 0.86 BTK (0.79) BTKEGFRKDRERBB4ERBB2
SCHEMBL17683823 0.85 EGFR (0.72) BTKAURKBAURKAEGFRERBB4
SCHEMBL17683789 0.82 BTK (1.00) BTKEGFRKDRERBB4ERBB2
SCHEMBL17675298 0.78 EGFR (0.67) BTKEGFRERBB4ERBB2MAPK14
SCHEMBL17675224 0.78 EGFR (0.70) BTKAURKBAURKAEGFRERBB4
SCHEMBL17675188 0.77 EGFR (0.74) BTKAURKBAURKAEGFRERBB2
SCHEMBL8933899 0.76 AURKB (0.94) AURKBAURKAEGFRKDRMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016055982-A1 QUINOLINE AND QUINAZOLINE COMPOUNDS ACERTA PHARMA B.V. (NL) 2016-04-14 WO claimed