SCHEMBL17675602

SCHEMBL17675602

CC#CC(=O)Nc1cc2c(Nc3ccc(C(=O)Nc4ccccn4)cc3)ccnc2cc1OC

nearest known ligand 0.76

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BTK Q06187 11/20 0.76
EGFR P00533 9/20 0.63
TEC P42680 2/20 0.55
TXK P42681 2/20 0.55
BLK P51451 2/20 0.55
BMX P51813 2/20 0.55
ERBB4 Q15303 2/20 0.55
ERBB2 P04626 2/20 0.55
JAK3 P52333 1/20 0.55
ITK Q08881 1/20 0.55
PDGFRA P16234 1/20 0.48
DNMT1 P26358 2/20 0.47
DNMT3L Q9UJW3 1/20 0.46
DNMT3A Q9Y6K1 1/20 0.46
F2 P00734 1/20 0.46
AURKA O14965 1/20 0.44
AURKB Q96GD4 1/20 0.44
KDR P35968 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17675397 0.89 BTK (0.70) BTKEGFRERBB4ERBB2AURKA
SCHEMBL17683789 0.86 BTK (1.00) BTKEGFRTECTXKBLK
SCHEMBL17675184 0.86 BTK (0.73) BTKEGFRDNMT1DNMT3LDNMT3A
SCHEMBL17683840 0.82 BTK (0.79) BTKEGFRTECTXKBLK
SCHEMBL17675586 0.79 EGFR (0.62) BTKEGFRTECTXKBLK
SCHEMBL17675255 0.79 BTK (0.85) BTKEGFRTECTXKBLK
SCHEMBL17675187 0.78 DNMT1 (0.66) BTKEGFRDNMT1DNMT3LDNMT3A
SCHEMBL17675217 0.78 KDR (0.63) BTKEGFRERBB2AURKAAURKB
SCHEMBL17675558 0.77 BTK (0.82) BTKEGFRTECTXKBLK
SCHEMBL17683763 0.77 BTK (1.00) BTKEGFRTECTXKBLK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016055982-A1 QUINOLINE AND QUINAZOLINE COMPOUNDS ACERTA PHARMA B.V. (NL) 2016-04-14 WO claimed