SCHEMBL17675452

SCHEMBL17675452

O=C(Nc1ccccn1)c1ccc(Oc2ccnc3cc(OCCOC4CCCCO4)c([N+](=O)[O-])cc23)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 15/20 0.52
TEC P42680 2/20 0.49
TXK P42681 2/20 0.49
BLK P51451 2/20 0.49
BMX P51813 2/20 0.49
ERBB4 Q15303 2/20 0.49
EGFR P00533 11/20 0.48
ERBB2 P04626 1/20 0.47
JAK3 P52333 1/20 0.47
ITK Q08881 1/20 0.47
KDR P35968 2/20 0.41
PDGFRA P16234 2/20 0.41
CYP3A4 P08684 1/20 0.41
KIT P10721 1/20 0.39
AXL P30530 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17675478 0.85 BTK (0.60) BTKTECTXKBLKBMX
SCHEMBL17675573 0.83 BTK (0.55) BTKTECTXKBLKBMX
SCHEMBL17675543 0.82 BTK (0.62) BTKTECTXKBLKBMX
SCHEMBL17675464 0.82 BTK (0.71) BTKTECTXKBLKBMX
SCHEMBL17675287 0.81 BTK (0.61) BTKTECTXKBLKBMX
SCHEMBL17675309 0.81 BTK (0.65) BTKTECTXKBLKBMX
SCHEMBL17675210 0.80 BTK (0.67) BTKTECTXKBLKBMX
SCHEMBL17675365 0.78 BTK (0.59) BTKTECTXKBLKBMX
SCHEMBL17675501 0.78 BTK (0.57) BTKTECTXKBLKBMX
SCHEMBL17675318 0.73 BTK (0.66) BTKTECTXKBLKBMX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016055982-A1 QUINOLINE AND QUINAZOLINE COMPOUNDS ACERTA PHARMA B.V. (NL) 2016-04-14 WO disclosed