SCHEMBL17679934

SCHEMBL17679934

C#Cc1ccc(C#N)cc1CC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.44
EGLN2 Q96KS0 1/20 0.39
ABCC9 O60706 1/20 0.38
ABCC8 Q09428 1/20 0.38
KCNJ11 Q14654 1/20 0.38
KCNJ8 Q15842 1/20 0.38
TRPV4 Q9HBA0 1/20 0.36
PGR P06401 1/20 0.36
ALDH1A1 P00352 1/20 0.34
GSK3B P49841 2/20 0.34
IMPDH2 P12268 1/20 0.34
IMPDH1 P20839 1/20 0.34
DRD2 P14416 1/20 0.34
DRD3 P35462 1/20 0.34
SETDB1 Q15047 1/20 0.34
ELANE P08246 1/20 0.33
LOXL2 Q9Y4K0 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23018392 0.86 CYP2A6 (0.48) CYP2A6EGLN2ABCC9ABCC8KCNJ11
SCHEMBL17679940 0.85 CYP2A6 (0.39) CYP2A6EGLN2ABCC9ABCC8KCNJ11
SCHEMBL13824727 0.78 CYP2A6 (0.52) CYP2A6EGLN2ABCC9ABCC8KCNJ11
SCHEMBL2934457 0.77 CYP2A6 (0.47) CYP2A6EGLN2ABCC9ABCC8KCNJ11
SCHEMBL12910016 0.76 CYP2A6 (0.47) CYP2A6EGLN2ABCC9ABCC8KCNJ11
SCHEMBL2154388 0.76 EGLN2 (0.52) CYP2A6EGLN2ABCC9ABCC8KCNJ11
SCHEMBL12959691 0.75 PDE3B (0.35) CYP2A6ALDH1A1MEN1KMT2A
SCHEMBL17530142 0.75 MAPT (0.36) CYP2A6ALDH1A1
SCHEMBL11661685 0.75 TRPA1 (0.39) CYP2A6ALDH1A1
SCHEMBL13199458 0.75 CYP2A6 (0.48) CYP2A6EGLN2ABCC9ABCC8KCNJ11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016055947-A1 ALKYNE COMPOUNDS AS S-NITROSOGLUTATHIONE REDUCTASE INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2016-04-14 WO disclosed