SCHEMBL17680285

SCHEMBL17680285

CC(C)(N)c1ccc(-c2cccnc2)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.73
CYP2A6 P11509 5/20 0.56
CYP3A4 P08684 3/20 0.56
ALDH1A1 P00352 1/20 0.56
CYP1A2 P05177 1/20 0.56
MKNK1 Q9BUB5 4/20 0.50
MKNK2 Q9HBH9 4/20 0.50
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA9 Q16790 1/20 0.50
AKT1 P31749 1/20 0.49
AKT2 P31751 1/20 0.49
CYP11B2 P19099 1/20 0.49
GPR55 Q9Y2T6 1/20 0.48
NPC1 O15118 1/20 0.47
CYP19A1 P11511 2/20 0.47
DGAT1 O75907 1/20 0.47
KCNH2 Q12809 1/20 0.47
CYP2C9 P11712 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL31303016 0.98 KIF11 (0.71) KIF11CYP2A6CYP3A4ALDH1A1CYP1A2
SCHEMBL23666164 0.85 KIF11 (1.00) KIF11CYP2A6CYP3A4ALDH1A1CYP1A2
SCHEMBL1623940 0.85 KIF11 (1.00) KIF11CYP2A6CYP3A4ALDH1A1CYP1A2
SCHEMBL4502483 0.81 KIF11 (0.73) KIF11CYP2A6CYP3A4ALDH1A1CYP1A2
SCHEMBL29468037 0.81 NPC1 (0.68) KIF11CYP2A6CYP3A4ALDH1A1CYP1A2
SCHEMBL6552315 0.81 NPC1 (0.68) KIF11CYP2A6CYP3A4ALDH1A1CYP1A2
SCHEMBL22778182 0.81 NPC1 (0.68) KIF11CYP2A6CYP3A4ALDH1A1CYP1A2
SCHEMBL25390854 0.80 KIF11 (0.78) KIF11CYP2A6CYP3A4ALDH1A1CYP1A2
SCHEMBL24534338 0.79 CYP2A6 (0.88) KIF11CYP2A6CYP3A4ALDH1A1CYP1A2
SCHEMBL29360677 0.79 CYP2A6 (0.88) KIF11CYP2A6CYP3A4ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024258789-A1 MODULATORS OF CDK2 AND USES THEREOF TRIANA BIOMEDICINES, INC. (US) 2024-12-19 WO disclosed
US-20170247336-A1 SUBSTITUTED PYRIMIDINES AS INHIBITORS OF HIF PROLYL HYDROXYLASE MERCK SHARP & DOHME CORP. (US) 2017-08-31 US disclosed
US-20170247336-A1 SUBSTITUTED PYRIMIDINES AS INHIBITORS OF HIF PROLYL HYDROXYLASE MERCK SHARP & DOHME CORP. (US) 2017-08-31 US disclosed
US-20170247336-A1 SUBSTITUTED PYRIMIDINES AS INHIBITORS OF HIF PROLYL HYDROXYLASE MERCK SHARP & DOHME CORP. (US) 2017-08-31 US disclosed
WO-2016057762-A1 SUBSTITUTED PYRIMIDINES AS INHIBITORS OF HIF PROLYL HYDROXYLASE MERCK SHARP & DOHME CORP (US) 2016-04-14 WO disclosed
WO-2016054804-A1 SUBSTITUTED PYRIMIDINES AS INHIBITORS OF HIF PROLYL HYDROXYLASE MERCK SHARP & DOHME CORP. (US) 2016-04-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170247336-A1 SUBSTITUTED PYRIMIDINES AS INHIBITORS OF HIF PROLYL HYDROXYLASE HIF1AN, HIF1A, EGLN2 KIF11 4607/4885CYP2A6 778/4885CYP3A4 2126/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.