SCHEMBL17680468

SCHEMBL17680468

Cc1nc(CNC(=O)OC(C)(C)C)ccc1Br

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.44
CA2 P00918 4/20 0.44
CA9 Q16790 4/20 0.44
CA12 O43570 3/20 0.44
KDM4A O75164 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.40
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
IGF1R P08069 1/20 0.38
LCK P06239 2/20 0.38
NAMPT P43490 1/20 0.38
BCHE P06276 1/20 0.38
CACNA1H O95180 1/20 0.37
CACNA1B Q00975 1/20 0.37
CACNA1C Q13936 1/20 0.37
CYP1A2 P05177 1/20 0.37
DYRK1A Q13627 1/20 0.37
CA4 P22748 1/20 0.37
CA7 P43166 1/20 0.37
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31104352 1.00 CA1 (0.44) CA1CA2CA9CA12KDM4A
SCHEMBL8218002 0.87 CA12 (0.45) CA1CA2CA9CA12KDM4A
SCHEMBL31103954 0.84 CA1 (0.45) CA1CA2CA9CA12KDM4A
SCHEMBL8223789 0.84 CA1 (0.42) CA1CA2CA9CA12KDM4A
SCHEMBL31432404 0.83 CA12 (0.44) CA1CA2CA9CA12KDM4A
SCHEMBL31380377 0.79 KDM4A (0.45) CA1CA12KDM4ABCHECYP1A2
SCHEMBL29664294 0.79 KDM4A (0.44) CA1CA2CA9CA12KDM4A
SCHEMBL26697003 0.79 NPSR1 (0.47) CA1CA2CA9CA12KDM4A
SCHEMBL31380399 0.78 MEN1 (0.44) CA1CA2CA9CA12KDM4A
SCHEMBL533745 0.78 RAB9A (0.34) LMNAIGF1RMEN1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016054807-A1 TrkA KINASE INHIBITORS, COMPOSITIONS AND METHODS THEREOF MERCK SHARP & DOHME CORP. (US) 2016-04-14 WO disclosed