SCHEMBL1768286

SCHEMBL1768286

Cc1c(OC2CCN(C(=O)OC3(C)CC3)CC2F)ncnc1N1CCn2nccc21

nearest known ligand 0.39

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 19/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13965575 1.00 GPR119 (0.39) GPR119CYP2C9CYP2C19
SCHEMBL12649747 1.00 GPR119 (0.39) GPR119CYP2C9CYP2C19
SCHEMBL13836355 0.89 PIK3CD (0.41) GPR119
SCHEMBL1768120 0.89 PIK3CD (0.41) GPR119
SCHEMBL12649728 0.89 PIK3CD (0.41) GPR119
SCHEMBL13836938 0.87 PIK3CD (0.34) GPR119
SCHEMBL1768164 0.87 PIK3CD (0.34) GPR119
SCHEMBL13836721 0.87 PIK3CD (0.34) GPR119
SCHEMBL13965574 0.87 GPR119 (0.44) GPR119CYP2C9
SCHEMBL1768324 0.87 GPR119 (0.44) GPR119CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2504342-A1 IMIDAZO-PYRAZOLES AS GPR119 INHIBITORS Pfizer Inc. (US) 2012-10-03 EP claimed
WO-2011061679-A1 IMIDAZO-PYRAZOLES AS GPR119 INHIBITORS PFIZER INC. (US) 2011-05-26 WO claimed