SCHEMBL17687

SCHEMBL17687

Nc1ccc(S(=O)(=O)C#CCN2CCN(c3ccc(C(O)(C(F)(F)F)C(F)(F)F)cc3)CC2)cn1

nearest known ligand 0.66

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GCK P35557 20/20 0.66
GCKR Q14397 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16932 0.91 GCK (0.67) GCKGCKR
SCHEMBL18383 0.91 GCK (0.67) GCKGCKR
SCHEMBL16675 0.91 GCK (0.67) GCKGCKR
SCHEMBL15576170 0.90 GCK (0.53) GCKGCKR
SCHEMBL15575148 0.88 GCKR (0.53) GCKGCKR
SCHEMBL15575275 0.88 GCKR (0.54) GCKGCKR
SCHEMBL15575336 0.88 GCKR (0.54) GCKGCKR
SCHEMBL15575586 0.87 GCKR (0.55) GCKGCKR
SCHEMBL15575124 0.87 GCKR (0.58) GCKGCKR
SCHEMBL15201251 0.85 GCK (0.52) GCKGCKR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013123444-A1 SULFONYL COMPOUNDS THAT INTERACT WITH GLUCOKINASE REGULATORY PROTEIN AMGEN INC. (US) 2013-08-22 WO disclosed
EP-2609081-A1 SULFONYLPIPERAZINE DERIVATIVES THAT INTERACT WITH GLUCOKINASE REGULATORY PROTEIN FOR THE TREATMENT OF DIABETES Amgen Inc. (US) 2013-07-03 EP disclosed
WO-2012027261-A1 SULFONYLPIPERAZINE DERIVATIVES THAT INTERACT WITH GLUCOKINASE REGULATORY PROTEIN FOR THE TREATMENT OF DIABETES AMGEN INC. (US) 2012-03-01 WO disclosed