SCHEMBL17689149

SCHEMBL17689149

Cc1ccc(-c2ncco2)cc1S(C)(=O)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.42
EDNRB P24530 5/20 0.40
EDNRA P25101 5/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA12 O43570 1/20 0.40
CA9 Q16790 1/20 0.40
BRD4 O60885 2/20 0.39
IL2 P60568 1/20 0.39
LTA4H P09960 1/20 0.39
NR1H2 P55055 1/20 0.39
NR1H3 Q13133 1/20 0.39
CA4 P22748 1/20 0.38
CA7 P43166 1/20 0.38
PIK3CD O00329 1/20 0.38
PIK3CG P48736 1/20 0.38
ACLY P53396 1/20 0.37
BRD2 P25440 1/20 0.37
BRD3 Q15059 1/20 0.37
P2RX7 Q99572 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17689125 0.84 EDNRA (0.39) EDNRBEDNRABRD4LTA4HACLY
SCHEMBL18230068 0.81 PIK3CD (0.40) EDNRBEDNRABRD4IL2LTA4H
SCHEMBL18229961 0.81 BRD4 (0.38) EDNRBEDNRABRD4LTA4HPIK3CD
SCHEMBL18930006 0.79 NPC1 (0.46) BRD4IL2LTA4HP2RX7HPGDS
SCHEMBL8591966 0.76 LTA4H (0.47) EDNRBEDNRALTA4HHPGDS
SCHEMBL4764672 0.74 LTA4H (0.42) EDNRBEDNRABRD4IL2LTA4H
SCHEMBL10317579 0.74 NPC1 (0.51) BRD4IL2LTA4HP2RX7HPGDS
SCHEMBL377220 0.74 IL2 (0.46) BRD4IL2LTA4HP2RX7HPGDS
SCHEMBL6499200 0.74 NPC1 (0.50) BRD4IL2LTA4HP2RX7HPGDS
SCHEMBL1459892 0.74 NPC1 (0.44) BRD4IL2LTA4HP2RX7HPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2922841-B1 ALKYL-AMIDE-SUBSTITUTED PYRIDYL COMPOUNDS USEFUL AS MODULATORS OF IL-12, IL-23 AND/OR IFN ALPHA RESPONSES BRISTOL MYERS SQUIBB CO (US) 2017-06-07 EP disclosed
US-9315494-B2 Alkyl-amide-substituted pyridyl compounds useful as modulators of IL-12, IL-23 and/or IFNα responses BRISTOL-MYERS SQUIBB COMPANY (US) 2016-04-19 US disclosed