SCHEMBL1768930

SCHEMBL1768930

CN(C)c1ccc(C(F)(F)F)cc1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 3/20 0.49
PDK2 Q15119 2/20 0.42
NR1H3 Q13133 2/20 0.41
PTGS2 P35354 2/20 0.40
PTGS1 P23219 1/20 0.40
MRGPRX4 Q96LA9 1/20 0.39
HTR2A P28223 1/20 0.39
SLC6A4 P31645 1/20 0.39
KCNH2 Q12809 1/20 0.39
MAPT P10636 2/20 0.39
ALDH1A1 P00352 1/20 0.39
NR1H2 P55055 1/20 0.38
CYP2D6 P10635 1/20 0.38
HTT P42858 1/20 0.38
GAA P10253 2/20 0.38
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
KDM4E B2RXH2 1/20 0.38
IDH2 P48735 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27766668 0.84 MAPT (0.47) PDE2APTGS2HTR2ASLC6A4KCNH2
SCHEMBL12401761 0.82 CYP2C19 (0.40) NR1H3PTGS2PTGS1KCNH2MAPT
SCHEMBL170653 0.79 ESR1 (0.49) PDE2AMAPTCYP2D6GAAIDH2
SCHEMBL8346846 0.79 PDK2 (0.51) PDE2APDK2NR1H3MRGPRX4MAPT
SCHEMBL11544632 0.78 ALDH1A1 (0.46) PDE2APDK2NR1H3MAPTALDH1A1
SCHEMBL18160746 0.78 IDH2 (0.38) PDE2ACYP2D6GAAIDH2KMT2A
SCHEMBL17993800 0.76 ALDH1A1 (0.37) PDE2ASLC6A4MAPTALDH1A1CYP2D6
SCHEMBL2968966 0.76 GAA (0.50) SLC6A4MAPTALDH1A1GAALMNA
SCHEMBL5108912 0.76 KDM4E (0.44) PDE2APDK2NR1H3MRGPRX4MAPT
SCHEMBL13696457 0.73 KDM1A (0.40) PDE2AMAPTCYP2D6GAAIDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111039792-B Preparation method of aniline compound 苏州开元民生科技股份有限公司 2022-10-14 CN claimed
CN-117777024-A Improved process for preparing arylpyrazole nitriles 江苏优普生物化学科技股份有限公司 2024-03-29 CN disclosed
CN-111039792-B Preparation method of aniline compound 苏州开元民生科技股份有限公司 2022-10-14 CN disclosed
CN-111039792-B Preparation method of aniline compound 苏州开元民生科技股份有限公司 2022-10-14 CN disclosed
CN-216321856-U Device for recovering dimethylamine in process of synthesizing fipronil 山东海利尔化工有限公司 2022-04-19 CN disclosed
CN-110845340-B Preparation method of fipronil intermediate 苏州开元民生科技股份有限公司 2022-03-22 CN disclosed
WO-2011058577-A1 PROCESS FOR SYNTHESIZING POLYHALOGENATED PERHALOALKYLANILINE COMPOUNDS GHARDA KEKI HORMUSJI (IN) 2011-05-19 WO disclosed
CN-1436769-A Prepn process of 2,6-dichloro-4-trifluoro methylaniline SHANGHAI TIANHAO MEDICINE SCI (CN) 2003-08-20 CN disclosed
US-5616810-A DEALKYLATION BY REACTING AN N-ALKYL OF N,N-DIALKYL ANILINE WITH AMMONIA OR A PRIMARY OR SECONDARY AMINE USING A PYRIDINE SALT CATALYST RHONE-POULENC CHIMIE (FR) 1997-04-01 US disclosed
US-5401882-A Reaction of halobenzenes with dialkyl amide to form dialkyl anilines, dealkylation RHONE-POULENC CHIMIE (FR) 1995-03-28 US disclosed