SCHEMBL17690652

SCHEMBL17690652

CCc1nc(C(N)=O)c(Nc2ccc(N3CCC(N4CCN(C)CC4)CC3)cc2)nc1NC1CCCCCC1

nearest known ligand 0.86

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EML4 Q9HC35 16/20 0.86
ALK Q9UM73 16/20 0.86
RET P07949 12/20 0.86
ROS1 P08922 12/20 0.86
FLT3 P36888 12/20 0.86
EGFR P00533 2/20 0.67
BMPR1B O00238 1/20 0.67
PLK4 O00444 1/20 0.67
CIT O14578 1/20 0.67
AURKA O14965 1/20 0.67
GAK O14976 1/20 0.67
EPHB6 O15197 1/20 0.67
RIPK2 O43353 1/20 0.67
BUB1 O43683 1/20 0.67
SNRNP200 O75643 1/20 0.67
STK16 O75716 1/20 0.67
STK10 O94804 1/20 0.67
MAP4K4 O95819 1/20 0.67
LATS1 O95835 1/20 0.67
SLC25A5 P05141 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL282960 0.93 RET (1.00) EML4ALKRETROS1FLT3
SCHEMBL282459 0.93 EML4 (1.00) EML4ALKRETROS1FLT3
SCHEMBL282458 0.93 EML4 (1.00) EML4ALKRETROS1FLT3
SCHEMBL16206860 0.91 EML4 (0.76) EML4ALKRETROS1FLT3
SCHEMBL16206865 0.91 EML4 (0.76) EML4ALKRETROS1FLT3
SCHEMBL16195726 0.90 EML4 (0.76) EML4ALKRETROS1FLT3
SCHEMBL16195564 0.90 EML4 (0.75) EML4ALKRETROS1FLT3
SCHEMBL16206870 0.90 EML4 (0.75) EML4ALKRETROS1FLT3
SCHEMBL10129857 0.89 RET (0.94) EML4ALKRETROS1FLT3
SCHEMBL16207089 0.88 EGFR (0.77) EML4ALKRETROS1FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3009428-A1 DIAMINO HETEROCYCLIC CARBOXAMIDE COMPOUND Astellas Pharma Inc. (JP) 2016-04-20 EP disclosed