SCHEMBL17690946

SCHEMBL17690946

Bc1cnn2c(NC(=O)OC(C)(C)C)cc(N3CCCN(C(=O)OC(C)(C)C)CC3)nc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CKS1B P61024 2/20 0.49
SKP1 P63208 2/20 0.49
SKP2 Q13309 2/20 0.49
GALR2 O43603 1/20 0.43
GALR1 P47211 1/20 0.43
MAPT P10636 2/20 0.40
MAP4K4 O95819 1/20 0.40
PTPN11 Q06124 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CDK2 P24941 1/20 0.39
TSHR P16473 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
P2RX3 P56373 1/20 0.39
PDE10A Q9Y233 1/20 0.39
LRRK2 Q5S007 1/20 0.38
GPR119 Q8TDV5 2/20 0.38
TBK1 Q9UHD2 1/20 0.38
WNT3A P56704 1/20 0.38
MET P08581 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14413677 0.90 CKS1B (0.48) CKS1BSKP1SKP2GALR2GALR1
SCHEMBL14413660 0.85 CKS1B (0.45) CKS1BSKP1SKP2GALR2GALR1
SCHEMBL14050908 0.80 TYK2 (0.39) CKS1BSKP1SKP2GALR2GALR1
SCHEMBL14050806 0.76 JAK3 (0.38) CKS1BSKP1SKP2GALR2GALR1
SCHEMBL14051003 0.74 CKS1B (0.49) CKS1BSKP1SKP2GALR2GALR1
SCHEMBL20533951 0.72 HPGD (0.40) CKS1BSKP1SKP2MAPTMEN1
SCHEMBL24851168 0.72 CKS1B (0.53) CKS1BSKP1SKP2GALR2GALR1
SCHEMBL14413674 0.72 CKS1B (0.51) CKS1BSKP1SKP2CDK2PDE10A
SCHEMBL1934892 0.72 CSNK2B (0.51) CKS1BSKP1SKP2MAPTMAP4K4
SCHEMBL24851476 0.72 CKS1B (0.55) CKS1BSKP1SKP2GALR2GALR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1931677-B1 NOVEL PYRAZOLOPYRIMIDINES AS CYCLIN DEPENDENT KINASE INHIBITORS MERCK SHARP & DOHME (US) 2016-04-20 EP disclosed