SCHEMBL17707486

SCHEMBL17707486

O=C1Cc2cc(C(=O)C3(Cc4ccccc4)CCN(C(=O)O)C3)ccc2N1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 3/20 0.51
HTR1A P08908 1/20 0.44
DRD2 P14416 1/20 0.44
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
HTR7 P34969 1/20 0.44
DRD3 P35462 1/20 0.44
HTR2B P41595 1/20 0.44
SMYD3 Q9H7B4 10/20 0.43
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
HSD11B1 P28845 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL441501 0.88 CRBN (0.51) GRIN2BHTR1ADRD2HTR2AHTR2C
SCHEMBL415385 0.85 GRIN2B (0.47) GRIN2BHTR1ADRD2HTR2AHTR2C
SCHEMBL414839 0.82 SLC6A2 (0.59) GRIN2BHTR1ADRD2HTR2AHTR2C
Hydrochloric Acid SCHEMBL447045 0.81 SLC6A2 (0.58) GRIN2BHTR1ADRD2HTR2AHTR2C
SCHEMBL17707503 0.81 IP6K1 (0.40) HTR1AHTR2AHTR7SLC6A2SLC6A4
SCHEMBL17707505 0.80 SLC6A2 (0.42) HTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL1691802 0.77 SLC6A2 (0.70) SLC6A2SLC6A4SLC6A3
SCHEMBL1692154 0.74 SLC6A2 (0.44) SLC6A2SLC6A4SLC6A3
SCHEMBL12350482 0.74 SMYD3 (0.47) GRIN2BHTR1ADRD2HTR2AHTR2C
SCHEMBL8117852 0.73 GRIN2B (0.75) GRIN2BHTR1ADRD2HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2684871-B1 Heteroaryl pyrrolidinyl and piperidinyl ketone derivatives HOFFMANN LA ROCHE (CH) 2016-05-04 EP disclosed