SCHEMBL1692154

SCHEMBL1692154

Cn1ccc2cc(C(=O)C3(Cc4ccccc4)CCN(C(=O)O)C3)ccc21

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 7/20 0.44
SLC6A4 P31645 7/20 0.44
SLC6A3 Q01959 7/20 0.44
CYP2D6 P10635 2/20 0.44
KCNH2 Q12809 1/20 0.44
FAAH O00519 1/20 0.42
SCN5A Q14524 1/20 0.42
SCN9A Q15858 1/20 0.42
FASN P49327 1/20 0.41
CHRNA7 P36544 3/20 0.40
MAPK14 Q16539 1/20 0.38
MAOB P27338 1/20 0.38
OXTR P30559 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
F2 P00734 1/20 0.37
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL442532 0.88 SCN5A (0.40) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL415547 0.86 SLC6A2 (0.42) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL413425 0.83 SLC6A2 (0.61) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL413794 0.81 SLC6A2 (0.62) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL17707505 0.79 SLC6A2 (0.42) SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL1691802 0.78 SLC6A2 (0.70) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL443834 0.74 OPRD1 (0.38) SLC6A2SLC6A4SLC6A3HDAC6
SCHEMBL17707486 0.74 GRIN2B (0.51) SLC6A2SLC6A4SLC6A3
SCHEMBL415331 0.73 SLC6A2 (0.39) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL17707503 0.72 IP6K1 (0.40) SLC6A2SLC6A4SLC6A3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2297096-A2 ARYL KETONE AS MRI F. Hoffmann-La Roche AG (CH) 2011-03-23 EP disclosed
WO-2009153178-A2 ARYL KETONE AS MRI F. HOFFMANN-LA ROCHE AG (CH) 2009-12-23 WO disclosed