SCHEMBL17707489

SCHEMBL17707489

CCCC1(C(=O)c2cc3cc(F)ccc3n2S(=O)(=O)c2ccccc2)CCN(C(=O)O)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOD2 Q9HC29 3/20 0.44
NOD1 Q9Y239 3/20 0.44
HRH3 Q9Y5N1 1/20 0.41
PTGDR2 Q9Y5Y4 3/20 0.41
PTGDR Q13258 2/20 0.41
SLC2A1 P11166 1/20 0.41
ALOX5 P09917 1/20 0.38
ACLY P53396 1/20 0.37
ALDH1A1 P00352 3/20 0.36
USP2 O75604 1/20 0.36
CYP2C9 P11712 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HIF1A Q16665 1/20 0.36
HTT P42858 1/20 0.36
AVPR1A P37288 1/20 0.36
HDAC3 O15379 2/20 0.36
HDAC4 P56524 2/20 0.36
HDAC1 Q13547 2/20 0.36
HDAC7 Q8WUI4 2/20 0.36
HDAC2 Q92769 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL415416 0.92 NOD2 (0.45) NOD2NOD1HRH3PTGDR2PTGDR
SCHEMBL445020 0.89 NOD2 (0.42) NOD2NOD1HRH3PTGDR2PTGDR
SCHEMBL1972137 0.81 PTGDR2 (0.40) NOD2NOD1HRH3PTGDR2PTGDR
SCHEMBL10003942 0.73 NOD2 (0.78) NOD2NOD1PTGDR2PTGDRACLY
SCHEMBL413982 0.72 PTGDR (0.39) NOD2NOD1PTGDR2PTGDRSLC2A1
SCHEMBL442516 0.71 NR1H2 (0.40) NOD2NOD1HRH3PTGDR2PTGDR
SCHEMBL17707499 0.71 KMT2A (0.51) ALDH1A1LMNAKDM4EHPGDHSD17B10
SCHEMBL10003377 0.69 NOD2 (0.47) NOD2NOD1PTGDR2PTGDRSLC2A1
SCHEMBL3560737 0.68 PTGDR2 (0.53) NOD2NOD1PTGDR2PTGDRACLY
SCHEMBL443237 0.68 CYP2D6 (0.46) NOD2NOD1ALOX5ALDH1A1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2684871-B1 Heteroaryl pyrrolidinyl and piperidinyl ketone derivatives HOFFMANN LA ROCHE (CH) 2016-05-04 EP disclosed