SCHEMBL17707490

SCHEMBL17707490

O=C(O)N1CCCC1(Cc1ccccc1)C(=O)c1ccc2[nH]ccc2c1

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 8/20 0.61
SLC6A4 P31645 8/20 0.61
SLC6A3 Q01959 8/20 0.61
MAPK14 Q16539 2/20 0.50
CTNNB1 P35222 1/20 0.46
WNT3A P56704 1/20 0.46
ACHE P22303 1/20 0.46
HTR4 Q13639 1/20 0.46
SIGMAR1 Q99720 1/20 0.46
CYP2D6 P10635 2/20 0.44
CNR1 P21554 1/20 0.43
CNR2 P34972 1/20 0.43
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
KCNH2 Q12809 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL443408 0.87 SLC6A2 (0.53) SLC6A2SLC6A4SLC6A3MAPK14ACHE
SCHEMBL413879 0.84 SLC6A2 (0.57) SLC6A2SLC6A4SLC6A3MAPK14CTNNB1
SCHEMBL1691802 0.77 SLC6A2 (0.70) SLC6A2SLC6A4SLC6A3MAPK14CTNNB1
SCHEMBL414728 0.76 SLC6A2 (1.00) SLC6A2SLC6A4SLC6A3MAPK14CTNNB1
SCHEMBL442059 0.75 SLC6A2 (1.00) SLC6A2SLC6A4SLC6A3MAPK14CTNNB1
SCHEMBL413872 0.75 SLC6A2 (1.00) SLC6A2SLC6A4SLC6A3MAPK14CTNNB1
SCHEMBL413590 0.75 SLC6A2 (1.00) SLC6A2SLC6A4SLC6A3MAPK14CTNNB1
SCHEMBL413845 0.75 SLC6A2 (0.70) SLC6A2SLC6A4SLC6A3MAPK14CTNNB1
SCHEMBL707002 0.75 SIGMAR1 (0.43) ACHESIGMAR1L3MBTL1
SCHEMBL414749 0.74 SLC6A2 (1.00) SLC6A2SLC6A4SLC6A3MAPK14CTNNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2684871-B1 Heteroaryl pyrrolidinyl and piperidinyl ketone derivatives HOFFMANN LA ROCHE (CH) 2016-05-04 EP disclosed