SCHEMBL17713628

SCHEMBL17713628

Cc1cc(C)c(CNC(=O)c2csc(CCCC3CCC(N(C)C)CC3)c2C)c(=O)[nH]1

nearest known ligand 0.68

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EZH2 Q15910 20/20 0.68
EED O75530 16/20 0.68
RBBP4 Q09028 16/20 0.68
SUZ12 Q15022 16/20 0.68
AEBP2 Q6ZN18 16/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16212464 1.00 EZH2 (0.68) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL16212636 1.00 EZH2 (0.68) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL16213220 0.91 EED (0.64) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL20793077 0.90 EZH2 (0.71) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL16212973 0.90 EZH2 (0.65) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL16212562 0.89 EED (0.57) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL16212764 0.86 EED (0.60) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL17099641 0.86 EED (0.75) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL17099648 0.85 EED (0.71) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL17713684 0.84 EZH2 (0.55) EZH2EEDRBBP4SUZ12AEBP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3212639-A1 ENHANCER OF ZESTE HOMOLOG 2 INHIBITORS Glaxosmithkline Intellectual Property (No. 2) Limited (GB) 2017-09-06 EP claimed
WO-2016066697-A1 ENHANCER OF ZESTE HOMOLOG 2 INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED (GB) 2016-05-06 WO claimed
EP-3212639-A1 ENHANCER OF ZESTE HOMOLOG 2 INHIBITORS Glaxosmithkline Intellectual Property (No. 2) Limited (GB) 2017-09-06 EP disclosed
WO-2016066697-A1 ENHANCER OF ZESTE HOMOLOG 2 INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED (GB) 2016-05-06 WO disclosed